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4-fluoro-N-{2-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}benzamide
N4-[(1-benzyl-1H-imidazol-2-yl)methyl]-N4,5,6-trimethylpyrimidine-2,4-diamine
2,2-difluoro-N-[(2-methylphenyl)(pyridin-4-yl)methyl]propanamide
1-(2-chloropyridin-3-yl)-3-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}urea
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-(quinoxalin-6-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-({1-[(2,5-dimethylthiophen-3-yl)sulfonyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(5-ethylfuran-2-yl)methyl]piperidin-3-ol
6-chloro-2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-1,3-benzothiazole
2-ethyl-N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}pyrimidine-5-carboxamide
(3-{4-[(4-methoxy-2,3,6-trimethylphenyl)methyl]piperazin-1-yl}propyl)dimethylamine
5-cyclopropyl-N-ethyl-N-(pyridin-4-ylmethyl)-1-{4-[2-(trifluoromethyl)phenyl]pyrimidin-2-yl}-1H-pyrazole-4-carboxamide
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-(prop-2-en-1-yl)acetamide
5-[(4-benzylpiperidin-1-yl)methyl]-N-(oxolan-3-yl)-1,2-oxazole-3-carboxamide
N-methyl-5-phenyl-N-(quinolin-5-ylmethyl)-1,2-oxazole-3-carboxamide
1-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]azocane
2-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}pyrrolidin-2-yl)-1,3-benzothiazole
1'-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-cyclopropyl-3-(1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)propanamide
4-({2-[1-(2,3-dihydro-1H-indene-1-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(pent-4-enoyl)piperidine-4-carboxamide
2-{2-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenoxy}acetamide
2-[(5-acetylthiophen-3-yl)methyl]-7-cyclohexyl-2,7-diazaspiro[4.5]decan-6-one
6-methyl-4-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1,2-dihydropyridin-2-one
4-(hydroxymethyl)-5-methyl-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
methyl (1R,3S,3aR,6aS)-3-(3-acetyl-2,4,6-trimethylphenyl)-1,5-dimethyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
9-(4,6-dimethylpyrimidin-2-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
6-(furan-3-yl)-2-[3-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}butan-1-one
(1R,5R)-6-[3-(benzyloxy)propyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-(3-methoxyphenyl)-N-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-pyrazole-5-carboxamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyridin-2-ylmethyl)acetamide
2-cyclopentyl-N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}acetamide
N-[2-(4-{[3-(2H-1,3-benzodioxol-5-yl)propanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]oxolane-2-carboxamide
1-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]phenyl}-1H-1,2,4-triazole
1-{1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-4-yl}-2-phenylethan-1-ol
N-cyclopropyl-6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridazin-3-amine
1-({4-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)piperidin-4-ol
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-[4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
1-({5-[(2,6-difluoro-3-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
4-[1-(oxolan-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]-2-(propan-2-yl)pyrimidine
(1S,5R)-6-(cyclopropylmethyl)-3-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2,6-dimethoxy-N-[2-(pyridin-3-yl)ethyl]pyridine-3-carboxamide
5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
3-[(2-hydroxyethyl)({5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-yl})amino]-1λ6-thiolane-1,1-dione
4-(5-methyl-4-{[1-(thiophen-2-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carbonyl)-1,4-diazepane-1-carbaldehyde
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol
1-(2-chloroprop-2-en-1-yl)-3-[(ethylamino)methyl]-6,7-dimethoxy-1,2-dihydroquinolin-2-one