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1-(azepan-1-yl)-4-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)butane-1,4-dione
1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-3-methyl-2-(3-methylphenoxy)butan-1-one
2-amino-N-(2-methoxyethyl)-4-phenyl-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)[(1-methylpiperidin-2-yl)methyl]amine
N,N,5-trimethyl-4-{[3-(morpholin-4-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
methyl({[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
ethyl 5-({[4-(pyridin-3-yl)pyrimidin-2-yl]amino}methyl)furan-2-carboxylate
N4-({5,7-dimethylimidazo[1,2-a]pyridin-2-yl}methyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-benzyl-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-1,4-diazepan-6-ol
5-ethyl-6-methyl-2-[3-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
methyl 1-{3-[3-({[(4-fluorophenyl)methyl](methyl)amino}methyl)phenoxy]-2-hydroxypropyl}piperidine-4-carboxylate
2-(3-methylphenyl)-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridine
3-(4-fluorophenyl)-4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazin-2-one
5-(3-methylbutyl)-5-(piperidin-4-yl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
1-(3-methoxypropyl)-8-[1-(methylsulfanyl)propan-2-yl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}propan-1-ol
(4aS,7aR)-1-(1H-imidazol-2-ylmethyl)-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(dimethylamino)-1-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-2-(2-methylphenyl)ethan-1-one
4-ethyl-1-methyl-3-{1-[(1-phenyl-1H-pyrazol-5-yl)methyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(1-cyclohexylpiperidin-3-yl)methyl]-4-methyl-N-(pyridin-3-ylmethyl)-1H-imidazole-2-carboxamide
4-(5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)pyridine
(2S,4R)-1-[(2-chlorophenyl)methyl]-4-{[(2,5-dimethylphenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)propan-1-one
1-(3-methylbenzenesulfonyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
1-tert-butyl-4-({[(2-fluoro-4-methoxyphenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
(4aR,7aS)-4-(2-methoxypyrimidine-5-carbonyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
4-[5-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}methyl)thiophen-2-yl]-2-methylbut-3-yn-2-ol
N-methyl-N-(oxan-4-ylmethyl)-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
1-cyclopropyl-4-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyrrolidin-2-one
4-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}-2-(pyridin-4-yl)pyridine
3-(4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperazin-1-yl)-1λ6-thiolane-1,1-dione
N-[5-(4-benzylpiperidine-1-carbonyl)-2-(2-methoxyphenyl)-1-methyl-1H-1,3-benzodiazol-7-yl]acetamide
2-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-N,N-dimethylquinoline-4-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}thiophene-2-carboxamide
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-3-[4-(oxolane-2-carbonyl)piperazin-1-yl]propanamide
N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
1-{1-[(2E)-3-(2-chlorophenyl)prop-2-enoyl]piperidin-3-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
1-(1-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-1,4-diazepan-5-one
1-(3-methoxybenzoyl)-4-(2-methyl-1,3-thiazole-5-carbonyl)piperazine
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]pyridine-3-carboxamide
(3S,4R)-4-methyl-1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidine-3,4-diol
4-(1,3-benzothiazol-6-yl)-N-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-(furan-2-yl)-3-phenyl-N-(pyrimidin-4-ylmethyl)propanamide
{2-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]quinolin-3-yl}methanol
(3aR,6aR)-2-(2-methoxyethyl)-5-[3-(pyridin-4-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-fluoro-2-{6-oxa-9-azaspiro[4.5]decan-9-ylmethyl}quinolin-4-ol
(1-methyl-1H-imidazol-2-yl)(1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-4-yl)methanol
1-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]-4-(4-methoxyphenyl)butan-1-one