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1-methyl-5-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydropyridin-2-one
N-(3,5-dimethoxyphenyl)-3-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-3-yl}propanamide
3-({1-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]pyrrolidin-3-yl}methyl)benzoic acid
6-[4-(thiophen-2-ylmethyl)piperazin-1-yl]-9H-purine
2-methyl-1-[3-(3-phenylpropanoyl)piperidin-1-yl]-2-(pyrrolidin-1-yl)propan-1-one
3-fluoro-4-methoxy-N-[(1-methylpyrrolidin-3-yl)methyl]benzamide
1-methyl-3-(propan-2-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]-1H-pyrazole-5-carboxamide
N'-(5-chloro-2-methylphenyl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]propanediamide
(1R,5R)-6-benzyl-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-(3,3,5,5-tetramethylcyclohexyl)piperazin-2-yl}ethan-1-ol
4-[2-(1H-imidazol-2-yl)benzoyl]-N,N-dimethylpiperazine-1-carboxamide
3-(cyclopentylamino)-2-(thiophen-2-ylmethyl)propan-1-ol
3-[2-({[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-1,3-oxazolidin-2-one
2-(dimethylamino)-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(2-methylphenyl)acetamide
3-(2-hydroxyethyl)-1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[(1-methyl-1H-imidazol-2-yl)methyl]urea
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pentan-1-one
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}acetamide
1-(cyclobutylmethyl)-3-({[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
2-{5-[2-(butan-2-yl)phenoxymethyl]-3-methyl-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-[(3S,4R)-1-(1H-indazole-3-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
4-(furan-3-carbonyl)-3-methyl-1-phenylpiperazin-2-one
5-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxamide
2-chloro-4-[2-(3-cyanophenyl)-1H-imidazol-1-yl]benzoic acid
1-(1,1-dioxo-1λ6-thiolan-3-yl)-N-[(4-methylpyridin-2-yl)methyl]piperidine-4-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-ethyl-N-[2-(4-methylbenzenesulfonyl)ethyl]acetamide
(3S,9aR)-3-(4-aminobutyl)-8-(quinolin-6-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-cyclopropyl-4-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
3-(2-methoxyethyl)-1-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-3-(thiophen-3-ylmethyl)urea
4-amino-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-one
3-ethyl-4-[4-(3-hydroxy-3-methylbutyl)benzoyl]-1-methylpiperazin-2-one
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-(propan-2-yloxy)propanamide
4-methyl-5-{3-[5-(1-methyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]propyl}-1,3-thiazole
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
(3S,4R)-1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-4-methylpiperidine-3,4-diol
{[(3S,4R)-1-(3,5-difluoropyridine-2-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
4-ethanesulfonamido-N-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}benzamide
2-[2-(benzenesulfonyl)ethyl]-5-(dimethylamino)-2,3-dihydropyridazin-3-one
2-[1-(1-methylpiperidin-4-yl)-4-(1-phenylpiperidin-4-yl)piperazin-2-yl]ethan-1-ol
2-{3-cyclopropyl-5-[1-(pyrrolidin-1-yl)propan-2-yl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
9-(cyclopropylmethyl)-1-methyl-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-3-methylthiophene-2-carboxamide
3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}urea
4-[1-(4-chlorophenyl)-1H-pyrazol-4-yl]-N-[2-(morpholin-4-yl)ethyl]pyrimidin-2-amine
[(2S,4R)-4-(dimethylamino)-1-{[2-(methylamino)pyridin-3-yl]methyl}pyrrolidin-2-yl]methanol
N-(oxolan-2-ylmethyl)-5-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-ylmethyl}pyrimidin-2-amine
6-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]pyrimidin-4-amine
5-methanesulfonyl-N,2-dimethyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}pyrimidin-4-amine
N-methyl-2-(pyridin-3-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-2-(1H-1,2,4-triazol-3-yl)benzamide