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1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(phenylsulfanyl)ethan-1-one
N-{4-oxo-4-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]butan-2-yl}acetamide
N-(4-{[(1S,5R)-6-(cyclobutylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}phenyl)acetamide
1-(1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)-2-(1H-pyrazol-1-yl)ethan-1-one
1-(but-2-ynoyl)-N-[4-(3-fluorophenyl)phenyl]piperidine-3-carboxamide
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-1-(2-methoxyacetyl)piperidine-4-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(3-hydroxyphenyl)methyl]-N-methylpiperidine-3-carboxamide
N4-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-6-methylpyrimidine-2,4-diamine
4-[2-({4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethyl]benzene-1-sulfonamide
6-[(4aR,8aR)-7-cyclopentanecarbonyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2,4-dimethylpyridine-3-carbonitrile
1-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-3-methyl-3-phenylpiperidine
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
N-cycloheptyl-2-(1H-imidazol-2-yl)-N-(pyridin-3-ylmethyl)benzamide
1-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
7-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile
(4aS,7aR)-1-[(5-cyclopentylthiophen-2-yl)methyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
9-{[4-(2-aminoethyl)phenyl]methyl}-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-(2-methoxyphenoxy)azetidine
N-cyclopropyl-4-{[2-(6-hydroxypyrimidin-4-yl)ethyl]sulfamoyl}benzamide
{3-[(1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]phenyl}methanol
2-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridine-4-carboxamide
4-amino-2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methylphenyl]pyrimidine-5-carbonitrile
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(6-methylpyrimidin-4-yl)pyrrolidin-3-yl]methanol
4-(2-fluorophenyl)-2-{5-methyl-4-[4-(piperidin-1-yl)piperidine-1-carbonyl]-1H-pyrazol-1-yl}pyrimidine
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
2-cyclopropyl-6-oxo-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-1,6-dihydropyrimidine-5-carboxamide
3-[3-(propan-2-yloxy)benzoyl]-1-(1H-1,2,4-triazole-5-carbonyl)piperidine
6-cyclopropyl-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]pyrimidin-4-amine
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide
N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)-3-(2-methoxyphenyl)propanamide
N-{1-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]piperidin-4-yl}methanesulfonamide
3-methyl-1-(4,4,4-trifluorobutyl)-1,2-dihydroquinoxalin-2-one
4-(cyclopropylsulfamoyl)-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methylbenzamide
1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-phenylpiperazine
2-(furan-2-yl)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}azepane
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-3-amine
6-{3-[(3-chlorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyridine-2-carbonitrile
2-cyclopropyl-8-[2-(pyrrolidin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
8-benzyl-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(pyrazin-2-yl)ethyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
1-(morpholin-4-yl)-3-(3-{[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}phenoxy)propan-2-ol
N,N-diethyl-3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-[(2-methylpyridin-3-yl)oxy]-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidine-4-carboxylic acid
3-chloro-N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)benzamide
5-(2-{2-[(5-ethyl-2-methylpyrimidin-4-yl)amino]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
4-(3-{1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)-2,5-dimethylpyrimidine
(4-{[1-(3-ethoxybenzoyl)pyrrolidin-3-yl]methyl}phenyl)methanol
2-[3-(1H-imidazol-1-yl)pyrrolidin-1-yl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidine
4-{[1-(4-methylpiperazine-1-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
[(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl](methyl)[(3-methylthiophen-2-yl)methyl]amine