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7-{[1-(prop-2-en-1-yl)-1H-1,3-benzodiazol-2-yl]methyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-4-(4-ethoxy-3-methylphenyl)butan-1-one
4-{4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperazin-1-yl}-2-[1-(thiophen-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[3-(3-fluorophenyl)phenyl]-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidine-4-carboxamide
3-{[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-oxazolidin-2-one
N4,N4,5-trimethyl-N2-[1-(oxolan-2-ylmethyl)piperidin-4-yl]pyrimidine-2,4-diamine
ethyl 3-({1-[(4-chlorophenyl)methyl]-6-oxopiperidin-3-yl}formamido)propanoate
3-[(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)methyl]benzonitrile
4-methyl-6-(4-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperazin-1-yl)-2-propylpyrimidine
N-{2-[(4-chlorophenyl)methoxy]ethyl}-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
4-{[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}pyridine
N,7-dimethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-6-carboxamide
(2R,3R,6R)-5-[1-(methoxymethyl)cyclobutanecarbonyl]-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(5-ethylpyridin-2-yl)methyl]methylamine
(1S,5R)-3-benzyl-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-6-sulfonamide
3-[1-(1H-pyrazol-1-yl)propan-2-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
5-oxo-1-[4-(pyridin-2-yl)butyl]pyrrolidine-3-carboxylic acid
N-[(1R,3S)-3-{[3-(dimethylamino)propyl](methyl)carbamoyl}cyclopentyl]-1H-1,2,4-triazole-5-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(propan-2-yloxy)ethyl]benzamide
N-{[(2S,4S)-4-fluoro-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]pyrrolidin-2-yl]methyl}propanamide
6-(3-chlorophenyl)-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
1-cyclohexyl-5-[(2-methylphenyl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
N-methyl-N-(pyrimidin-4-ylmethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-(trifluoromethyl)pyrimidin-4-amine
4-(2,4-dioxoimidazolidin-1-yl)-N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]benzamide
2-(1,3-benzothiazol-2-ylmethyl)-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(4-methoxy-3-methylbenzoyl)piperidine
5-methoxy-3-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3,4-dihydroquinazolin-4-one
3-{[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
2-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}propanamide
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-[1-(thian-4-yl)piperidin-4-yl]acetamide
2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)-N-[2-(phenylsulfanyl)ethyl]-N-(prop-2-en-1-yl)acetamide
1-(1H-imidazole-2-carbonyl)-4-(oxan-4-yl)-1,4-diazepane-6-carboxylic acid
N-(2-hydroxyethyl)-N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-(4-methylphenyl)-N-{[5-(methylsulfanyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-(2,2-diphenylethyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3-[(2-fluorophenyl)formamido]-N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}propanamide
3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-5-methoxy-1,2-dimethyl-1H-indole
4-(4-fluorophenyl)-2-{[3-(furan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,3-thiazole
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[(1-ethyl-1H-pyrazol-3-yl)methyl]pyrrolidine-3-carboxylic acid
2-[benzyl({[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl})amino]ethan-1-ol
3-benzyl-5-{pyrazolo[1,5-a]pyridin-3-yl}-1H-1,2,4-triazole
1-{2-[3-(1-methyl-1H-pyrazol-3-yl)phenyl]phenyl}ethan-1-one
N-(1H-imidazol-2-ylmethyl)-3-propanamidobenzamide
(4aR,8aR)-4a-hydroxy-7-[6-hydroxy-2-(propan-2-yl)pyrimidin-4-yl]-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
methyl 2-[2-oxo-4-(quinoline-2-carbonyl)piperazin-1-yl]acetate
methyl 6-[3-(4-fluorophenoxymethyl)piperidin-1-yl]pyrimidine-4-carboxylate
methyl 5-[(1-acetylpiperidin-4-yl)amino]-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate