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2-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
3-methyl-9-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-3,9-diazaspiro[5.6]dodecane
3-[(2R,3R,6R)-5-[(1-propyl-1H-imidazol-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
(3S,5S)-1-(cyclopropylmethyl)-5-[(6-methylpyridin-3-yl)carbamoyl]piperidine-3-carboxylic acid
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-1-(methoxymethyl)cyclobutane-1-carboxamide
2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidin-4-ol
5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-2-(methylsulfanyl)pyrimidine
2-(1-benzothiophen-2-yl)-1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazole
2-(4-methylpiperazine-1-carbonyl)-1-(2-propyl-1,3-thiazole-4-carbonyl)piperazine
3-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide
13-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-methyl-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
methyl(1,2-oxazol-3-ylmethyl)[(4-{[1-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]amine
2-(1,2-oxazolidin-2-yl)-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
1-(2-aminoethyl)-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
3-(1-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}piperidin-4-yl)-1-(morpholin-4-yl)propan-1-one
(3R)-1-{[1-(naphthalen-2-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-ol
1-(3-chloro-5-fluorobenzoyl)-3-(1-ethyl-1H-imidazol-2-yl)piperidine
1-[5-(propan-2-yl)thiophene-3-carbonyl]pyrrolidin-3-ol
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-{4-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-1H-pyrazol-1-yl}acetamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2,5,6-trimethylpyrimidin-4-amine
7-(cyclohexylmethyl)-2-(pyridin-4-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
(2R,3R,6R)-5-cyclobutanecarbonyl-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{methyl[6-(4-methylthiophen-3-yl)pyridazin-3-yl]amino}ethan-1-ol
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}piperidin-4-amine
3-[(cyclopropylamino)methyl]-7-methyl-1-[(3-methylphenyl)methyl]-1,2-dihydroquinolin-2-one
2-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-2-azaspiro[4.4]nonane
1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
(2S)-N-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-methyl-N-[(3-methylthiophen-2-yl)methyl]acetamide
4-[7-(2,3-dichlorobenzoyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
3-(1,2-oxazinan-2-yl)-1-{3-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidin-1-yl}propan-1-one
(3R,4R)-4-ethyl-1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]piperidine-3,4-diol
1-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-2-(1-methyl-1H-imidazol-2-yl)piperidine
9-{[2-(ethylamino)pyrimidin-5-yl]methyl}-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
4-(methoxymethyl)-6-[3-(trifluoromethoxy)phenyl]pyrimidine
1-{3-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carbonyl]phenyl}-4-ethyl-3-methyl-1H-pyrazol-5-ol
4-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}morpholine-2-carboxamide
4-{1-azabicyclo[2.2.2]octan-3-yl}-N-(5-cyclobutyl-1,3,4-thiadiazol-2-yl)piperazine-1-carboxamide
N3,N3-bis(furan-2-ylmethyl)-N1,N1-dimethylpiperidine-1,3-dicarboxamide
2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-4-[(2-propyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
N-[2-(3-chlorophenyl)ethyl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-2-ethyl-N-(furan-2-ylmethyl)butanamide
1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
1-(azocan-1-yl)-3-{2-[(cyclobutylamino)methyl]-5-methoxyphenoxy}propan-2-ol
1-{2-methylthieno[3,2-d]pyrimidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
3-(6-hydroxy-6-methylheptan-2-yl)-1-[2-(methylsulfanyl)phenyl]urea
3-(3-methoxypropyl)-1-(3-methoxypyrazin-2-yl)piperidine-3-carboxylic acid
1-{1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-(3-methoxyphenyl)piperidine
3-(4-ethyl-1H-pyrazol-5-yl)-1-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]piperidine