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N1,N1-dimethyl-N3-{2-[(4-methylpyridin-2-yl)amino]ethyl}piperidine-1,3-dicarboxamide
N-[3-({[(1-cyclohexylpyrrolidin-3-yl)methyl]carbamoyl}amino)phenyl]acetamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
N-(4-fluoro-2-methylphenyl)-3-{1-[2-(methylsulfanyl)benzoyl]piperidin-3-yl}propanamide
N-(3-chloro-4-methoxyphenyl)-3-[1-(oxane-4-carbonyl)piperidin-3-yl]propanamide
N-({1-[(2E)-3-(5-chloro-2-hydroxyphenyl)-2-methylprop-2-en-1-yl]piperidin-3-yl}methyl)acetamide
3-phenoxy-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}azetidine
(1R,3S)-3-(2-hydroxyethoxy)-7-(5-methyl-1,3,4-thiadiazol-2-yl)-7-azaspiro[3.5]nonan-1-ol
4-(2H-1,3-benzodioxol-5-yloxy)-1-(3-methylpyrazin-2-yl)piperidine-4-carboxylic acid
4-{[2-(2,1,3-benzoxadiazol-4-yl)-1H-imidazol-1-yl]methyl}benzene-1-sulfonamide
2-(2-methylpropyl)-8-(pyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
ethyl 2-(4-{6-[ethyl(methyl)amino]pyrimidin-4-yl}piperazin-1-yl)acetate
1-(6-methylpyridin-2-yl)-4-(1-propylpiperidin-4-yl)piperazine
N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-3-hydroxy-1,2-oxazole-5-carboxamide
N-[4-(4-{[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]amino}piperidin-1-yl)phenyl]pyrazine-2-carboxamide
2-(adamantan-1-yl)-N-[1-(pyrazin-2-yl)piperidin-4-yl]acetamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-(pyrimidin-2-yl)pyrimidine
3-[2-(2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]-N-(2-ethylphenyl)propanamide
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-methoxyethyl)-4-{[(piperidin-4-ylmethyl)carbamoyl]amino}benzamide
(4aR,8aS)-1-[2-(2-methoxyphenyl)ethyl]-6-(thiophen-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
1-[4-(2-methoxypyridin-3-yl)phenyl]-2-(morpholin-4-yl)ethan-1-ol
4-hydroxy-2-{[(prop-2-en-1-yl)amino]methyl}quinoline-6-carboxamide
2-(3-fluorobenzenesulfonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[(2R,3R)-2-methoxy-1'-[3-(thiophen-2-yl)propanoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[(3-methylpyridin-4-yl)methyl]benzamide
2-(2-methoxyphenyl)-5-{1-[(2S)-1-methoxypropan-2-yl]-4-phenyl-1H-imidazol-5-yl}pyrimidine
2-(4-ethylpiperazin-1-yl)-N-(2-methylbutyl)-2,3-dihydro-1H-indene-2-carboxamide
3-amino-1-[2-methyl-2-(morpholin-4-ylmethyl)propyl]pyrrolidine-3-carboxylic acid
2-(2-{[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}ethyl)-1,2-dihydrophthalazin-1-one
3-[1-(4-chlorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]pyridazine
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}cyclopropan-1-amine
N,1-dimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
1-(3-methoxy-2-methylbenzoyl)-2-(4-methylpiperazine-1-carbonyl)piperazine
2-(2-{[methyl(2-methylpropyl)amino]methyl}phenyl)-6-(2-methylpropyl)-3,4-dihydropyrimidin-4-one
(3E)-N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}pent-3-enamide
4-(5-methylpyridin-2-yl)-1-(1,2,3,4-tetrahydroquinoline-8-carbonyl)piperidin-4-ol
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-3-methyl-1-(prop-2-en-1-yl)-1H-pyrazole
2-{4-[({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]phenyl}-6-methyl-3,4-dihydropyrimidin-4-one
8-(1H-indole-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[(2-amino-6-methylpyrimidin-4-yl)amino]-N-cyclohexylpropanamide
[3-(2-methoxyethyl)-1-(4-methyl-1H-imidazole-5-carbonyl)piperidin-3-yl]methanol
1-[2-({5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-yl}amino)ethyl]piperidin-3-ol
7-(2,4-dimethoxybenzenesulfonyl)-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[2-(3-chlorophenoxy)ethyl]-N-ethyl-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
4-[5-(2,6-dimethylpyrimidin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]benzene-1-sulfonamide
5-({methyl[(3-{2-[4-(pyridine-3-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amino}methyl)pyrrolidin-2-one
N-cyclopentyl-8-[2-(1H-imidazol-4-yl)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
4-{2-oxo-2-[(2S)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]ethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-methyl-N-(quinolin-5-ylmethyl)-1H-pyrazole-4-carboxamide