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2-(1-methylpiperidin-2-yl)-1-[4-(4-phenylpyrimidin-2-yl)piperazin-1-yl]ethan-1-one
N'-(3-ethylphenyl)-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]butanediamide
N-[2-(azepan-1-yl)ethyl]-N-(propan-2-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
2-[2-({2-cyclopropyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}methyl)phenoxy]acetic acid
ethyl 5-[4-(hydroxymethyl)phenyl]pyridine-3-carboxylate
3-(2-fluorophenyl)-1-[4-(pyridin-4-yl)piperidin-1-yl]propan-1-one
4-(2,5-dimethylbenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
[(3-fluorophenyl)methyl](methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-2-(thiophen-2-yl)ethan-1-one
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-(2-oxo-6-phenyl-1,2-dihydropyridine-3-carbonyl)piperidin-3-yl]propanoic acid
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl){[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}amine
N-benzyl-4-(1H-1,2,4-triazole-3-carbonyl)piperazine-1-sulfonamide
1-(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-3-yl)-4-(2-methoxyphenyl)piperazine
2-(2,4-difluorophenoxy)-1-[3-(3-methylphenoxy)azetidin-1-yl]ethan-1-one
N-[(3-ethoxy-4-methoxyphenyl)methyl]-1-[(2-fluorophenyl)methyl]piperidin-3-amine
{[(3S,4R)-1-(2-ethylpyrimidine-5-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
3-({1-[2-(pyridin-3-yl)acetyl]pyrrolidin-3-yl}methyl)benzamide
3-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]phenol
2-[(1S,5R)-3-[(2,6-dimethylphenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
5-(2H-1,3-benzodioxol-5-yl)-3-(3-methoxyphenoxymethyl)-1-methyl-1H-1,2,4-triazole
1-[(3-chloropyridin-4-yl)methyl]-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenyl)-6-(oxolan-3-yl)-3,4-dihydropyrimidin-4-one
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-({[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)piperidin-2-one
methyl (3aS,6aS)-2-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylate
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{[methyl(prop-2-yn-1-yl)amino]methyl}piperidin-2-one
1-cyclohexyl-2,6,6-trimethyl-3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indol-4-one
1-(4-chlorophenyl)-4-(1H-imidazol-2-ylmethyl)-5-methylpiperazin-2-one
(4aR,7aS)-1-ethyl-4-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(4-methoxyphenyl)-3-methyl-4-(morpholine-4-sulfonyl)piperazin-2-one
methyl 1-{[1-(2,2-dimethylpropyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}piperidine-4-carboxylate
2-({[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)pyrimidine
1-(6-oxo-1,6-dihydropyridazine-3-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
N-(3,3-dimethylbutyl)-5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
4-benzyl-3-ethyl-1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-1,4-diazepan-5-one
2-(dimethylamino)-7-(4-hydroxy-3-methylbenzoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{2-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}adamantane-1-carboxamide
7-(5-methylthiophen-2-yl)-4-(1H-1,2,4-triazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N,6-dimethyl-N-[4-(morpholin-4-yl)butyl]-4-oxo-4H-pyran-2-carboxamide
4-chloro-3-({[1-(1-methyl-1H-pyrazol-5-yl)propyl]carbamoyl}amino)-N-propylbenzamide
4-(1-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperidin-3-yl)morpholine
3-cyclopentyl-1-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)urea
{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}(methyl)[1-(pyridin-2-yl)ethyl]amine
1-[(4-chlorophenyl)methyl]-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperazine
2-(2-chloro-4-fluorophenoxymethyl)-N-[(1r,4r)-4-hydroxycyclohexyl]-1,3-oxazole-4-carboxamide
3-(furan-2-yl)-1-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}propan-1-one
1-[3-(3-fluorophenyl)benzoyl]-4-[2-(pyrrolidin-1-yl)ethyl]-1,4-diazepan-5-one
1-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)urea
5-{2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]acetyl}-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
6-({1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide