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ethyl 2-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-2-phenylacetate
ethyl 4-[(4-chlorophenyl)methyl]-1-(5-methylthiophene-2-carbonyl)piperidine-4-carboxylate
1-cyclopropanecarbonyl-4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1,4-diazepane
(1R,5R)-6-{[4-(2-hydroxyethoxy)phenyl]methyl}-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-(pentan-3-yl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(1S,5R)-3-(pyridin-3-ylmethyl)-6-(1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-chloro-N-{1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
3-(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidine-3-carbonyl)pyridine
9-(4-methoxy-3-methylbenzoyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-(4-methoxyphenyl)piperazine
2-cyclopropanecarbonyl-8-(3,5-dimethylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(3-ethoxy-4-methoxyphenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
1-(4-methoxyphenyl)-2,2-dimethyl-4-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperazine
methyl 2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]hexanoate
2-(cyclohex-1-en-1-yl)-N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)acetamide
1-[(3S,4S)-3-hydroxy-4-[4-(pyrimidin-2-yl)piperazin-1-yl]pyrrolidin-1-yl]-2-(methylsulfanyl)ethan-1-one
1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
3-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
N-[(1R,3R)-3-aminocyclopentyl]-2-[(3-methoxyphenyl)sulfanyl]acetamide
N-({7-[3-(2-chlorophenyl)propanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-fluorobenzamide
4-benzyl-3-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(5-methylthiophen-2-yl)sulfonyl]-3-[3-(trifluoromethyl)benzoyl]piperidine
1-[({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}carbamoyl)methyl]piperidine-4-carboxamide
3-(1H-imidazol-2-yl)-1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidine
1,5-dimethyl-4-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(2-propyl-1H-1,3-benzodiazol-1-yl)propanamide
2-ethyl-N-[(1-ethyl-1H-indazol-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N4-[2-(ethanesulfonyl)ethyl]-6-ethyl-5-methylpyrimidine-2,4-diamine
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(2-ethoxyphenyl)methyl]methylamine
4-[(2R)-3-hydroxy-2-methylpropyl]-1-(4-methoxyphenyl)piperazin-2-one
2-ethyl-4-({4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)pyrimidine
2-(4-fluorophenoxy)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
7-methoxy-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-(4-cyclohexylphenyl)-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1,2,4-triazin-3-amine
(4aS,8aR)-1-[2-(5-methylfuran-2-yl)ethyl]-6-(pyridin-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
5-{4-[1-(2-ethoxyethyl)-4-phenyl-1H-imidazol-5-yl]phenyl}pyrimidine
8-(3,5-dimethyl-1-benzofuran-2-carbonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[2-(dimethylamino)ethyl]-N-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
5-({4-[1-(dimethylamino)ethyl]piperidin-1-yl}methyl)-2-hydroxybenzoic acid
7-{2-[(4-methylpyridin-2-yl)amino]ethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-(pyridine-2-carbonyl)-8-azabicyclo[3.2.1]octane
(3R,4S)-4-cyclopropyl-1-[4-(diethylamino)benzoyl]pyrrolidin-3-amine
(4aR,7aS)-1-cyclopropanecarbonyl-4-(1-methyl-1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-1-(4-ethylpiperazin-1-yl)propan-1-one
2-(3-hydroxypropyl)-8-(4-methylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
3-(4-chlorophenyl)-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-sulfonamide
1-[(7-fluoroquinazolin-4-yl)amino]-3-(3-methoxyphenoxy)propan-2-ol
N-[1-(2-phenylethyl)piperidin-3-yl]-1,3-thiazole-4-carboxamide