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(5-{1-[(6-methoxypyridin-3-yl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidin-3-yl]urea
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
N4-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
3-chloro-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-6-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide
3-(1H-imidazol-1-yl)-1-[4-(3-methoxybenzoyl)piperazin-1-yl]propan-1-one
1-{[(2-fluoro-5-propanamidophenyl)carbamoyl]amino}cycloheptane-1-carboxamide
2-(1,4-dimethylpiperazin-2-yl)-N-[2-(3-phenoxyphenyl)ethyl]acetamide
4-(1-aminocyclobutanecarbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{2-oxa-7-azaspiro[4.5]decan-7-yl}-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
2-[4-(2-ethoxyethyl)piperazin-1-yl]pyrazine
4-[(2-methyl-1,3-thiazol-4-yl)methyl]-N-[3-(1H-pyrazol-5-yl)phenyl]piperazine-1-carboxamide
4-[7-(1-methyl-1H-pyrazole-5-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]thiomorpholine
N-(2H-1,3-benzodioxol-5-yl)-1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
(3aS,6aS)-2-cyclobutanecarbonyl-5-[(4-methyl-1,3-thiazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2,3-dimethyl-7-(morpholine-4-sulfonyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
3-(1H-indol-3-yl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}propanamide
4-[4-(3-methyl-1H-pyrazol-4-yl)phenyl]-1,3-thiazol-2-amine
1-ethyl-4-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
8-(2-propoxyacetyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{3-[(2-methoxyphenyl)methyl]-1-(6-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl}morpholine
1'-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]spiro[indene-1,4'-piperidine]
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
3-[1-(2-methanesulfonylethyl)-4-phenyl-1H-imidazol-5-yl]quinoline
1-methyl-5-{[(1-phenylcyclopentyl)methyl]amino}-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-amino-N-(2,1,3-benzoxadiazol-5-ylmethyl)-4-methyl-1,3-thiazole-5-carboxamide
(1R,5R)-6-benzyl-3-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
{2-[2-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]ethyl}dimethylamine
N-(dicyclopropylmethyl)-3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamide
7-hydroxy-4-(1H-indol-4-yl)-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
4-{[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]methyl}-2,1,3-benzoxadiazole
1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1,3-dimethyl-N-[2-(4-methylpiperazin-1-yl)butyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
8-(1,3-benzoxazol-2-yl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-1,8-diazaspiro[4.5]decane
3-[(1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)oxy]pyridine
(3R,4S)-1-(2-cyclopropylpyrimidine-5-carbonyl)-4-(propan-2-yl)pyrrolidin-3-amine
(5-{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
4-(pyridin-2-yl)-2-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrimidine
2-(2-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
(1S,5R)-3-[3-(2-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-3,9-diazabicyclo[3.3.2]decan-10-one
3-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-1-methyl-1,2-dihydroquinolin-2-one
2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]acetamide
N-butyl-2-(2,3-difluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]acetamide
1-(4-{[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)amino}piperidin-1-yl)ethan-1-one
(1S,5R)-3-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-3,9-diazabicyclo[3.3.2]decan-10-one
2-[3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazin-1-yl]ethan-1-ol
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[2-(methylsulfanyl)pyrimidin-4-yl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-methyl-1'-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one