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1-({5-[1-(2-amino-2-methylpropyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
(1R,3S)-3-amino-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}cyclohexane-1-carboxamide
2-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}benzoic acid
1-{2-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
(4aS,7aR)-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl (2S,4S,5R)-1,2-dimethyl-4-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]carbamoyl}-5-(2-methylphenyl)pyrrolidine-2-carboxylate
5-chloro-3-{4-[(1S,2S)-2-hydroxycyclohexyl]piperazine-1-carbonyl}-4,6-dimethyl-1,2-dihydropyridin-2-one
[(2S,6S)-4-(2-methylpyridin-4-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
4-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-1-ethyl-1,2-dihydropyridin-2-one
(3R,5R)-N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
4-(1H-1,3-benzodiazol-1-yl)-1-(6-methoxypyrimidin-4-yl)piperidine-4-carboxylic acid
2-(4-{[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]methyl}-2-methoxyphenoxy)acetamide
4-(3,5-difluoropyridine-2-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
(1R,5R)-6-(cyclobutylmethyl)-3-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2,1-benzoxazole-3-carboxamide
N-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-1-(1,3-benzothiazol-2-yl)piperidin-3-amine
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
2-(1-methyl-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-2-yl)ethan-1-ol
5-{3-oxo-3-[4-(pyridin-4-yl)piperidin-1-yl]propyl}imidazolidine-2,4-dione
2-(cyclohex-1-en-1-yl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}acetamide
methyl 2-(2-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}acetamido)-4-methyl-1,3-thiazole-5-carboxylate
1-(3-hydroxy-3-phenylpropyl)-1-methyl-3-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-{2-[(1-methylpiperidin-3-yl)methyl]-1H-1,3-benzodiazol-1-yl}acetamide
9-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidine
4-(hydroxymethyl)-1-{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}azepan-4-ol
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-5-[(methylsulfanyl)methyl]furan-2-carboxamide
2-methyl-8-(1H-pyrazol-1-yl)quinolin-4-ol
2-methyl-N-[1-(thiophen-2-yl)butyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-cyclopropyl-1-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]piperazine-2-carboxamide
2-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-1-ethyl-1H-1,3-benzodiazole
1-(3-cyano-4-ethoxyphenyl)-5-oxopyrrolidine-3-carboxylic acid
N-[(2S)-1-hydroxy-3-methylbutan-2-yl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5,5-diphenylpiperidin-2-one
N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(pyrimidin-4-ylmethyl)-1,3-oxazole-4-carboxamide
2-methyl-9-[(8-methylquinolin-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{[3-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}benzoic acid
3-{1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-1,3-oxazolidin-2-one
N-(4-cyano-2-ethylphenyl)-3-[(methylsulfanyl)methyl]piperidine-1-carboxamide
N-methyl-2-(1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}-3-oxopiperazin-2-yl)acetamide
N-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}-N,1-dimethylpiperidin-4-amine
8-({[1-(hydroxymethyl)cyclobutyl]methyl}amino)-2,6-dimethyloctan-2-ol
2-chloro-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-acetamidobenzamide
1-methyl-8-[3-(4-methylphenyl)propanoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
9-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(2R,3R,6R)-3-phenyl-5-(1,3-thiazol-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-4-(pyrrolidine-1-carbonyl)pyridine
1-amino-N-({1-[(6-chloropyridin-3-yl)methyl]pyrrolidin-3-yl}methyl)cyclopentane-1-carboxamide
4-{[(2S,4S)-2-[4-(adamantan-2-yl)piperazine-1-carbonyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidin-1-yl]methyl}quinoline