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2-methyl-6-{3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carbonyl}phenol
2-cyclopentyl-N-[(2-methylphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
(1S,5R)-6-(1H-indole-2-carbonyl)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-4-(piperidin-3-yl)benzamide
2-(2-methoxyethoxy)-1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
2-{4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-(1-carbamoylcyclopentyl)-3-phenyl-1H-pyrazole-4-carboxamide
N-(cyclopropylmethyl)-2-(3-methoxyphenyl)-N-(oxolan-2-ylmethyl)-1,3-benzoxazole-6-carboxamide
2-(methylsulfanyl)-N-[(3R,4S)-4-propyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]acetamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-2,9-diazaspiro[5.5]undecan-3-one
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(cyclohexylmethyl)methylamine
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(oxan-4-yl)ethyl]acetamide
4-[(5-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]-1,4-oxazepane
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[2-(5-methylthiophen-2-yl)ethyl]acetamide
[1-(2,3-dihydro-1H-inden-2-yl)-3-(3-methoxypropyl)piperidin-3-yl]methanol
2-amino-4-(1-ethyl-1H-pyrazol-4-yl)-7-hydroxy-5H,6H-benzo[h]quinoline-3-carbonitrile
ethyl 3-benzyl-1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidine-3-carboxylate
N-[1-(3-phenylpropyl)piperidin-3-yl]pyrrolidine-1-sulfonamide
5-(3,3-diphenylpiperidine-1-carbonyl)-1-methylpiperidin-2-one
N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-3-(2-oxoimidazolidin-1-yl)benzamide
[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](methyl){[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
2-{[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amino]methyl}pyridine-3-carboxylic acid
5-methyl-5-(4-methylpent-3-en-1-yl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}piperidin-2-one
4-(2-amino-3-cyano-6-cyclobutylpyridin-4-yl)-N-methylbenzene-1-sulfonamide
(2-methoxyethyl)(thiophen-2-ylmethyl){[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amine
2-methoxy-1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}ethan-1-one
3-[2-(2-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-1H-imidazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-methyl-N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-1,3-oxazole-4-carboxamide
1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
(2S)-N-[3-(4-fluorophenyl)phenyl]-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidine-2-carboxamide
3-(piperazine-1-carbonyl)-N-[2-(1,3-thiazol-2-yl)ethyl]benzene-1-sulfonamide
N-[(2-chlorophenyl)methyl]-N-(2-hydroxyethyl)-5-methyl-1,3-oxazole-4-carboxamide
1-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-2-[2-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)-4-phenylphenoxy]ethan-1-one
2-[4-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenyl]-3H,4H,5H,6H,7H,8H,9H-cyclohepta[d]pyrimidin-4-one
3-{2-[4-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}-4-(naphthalen-2-ylmethyl)piperazin-2-one
(5-{[5-(3-chlorophenyl)furan-2-yl]methyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
1-(2,3-dimethylphenyl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-amine
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidine
7-methyl-3-[1-(propan-2-yl)-1H-imidazol-2-yl]-1H-indole
2-(4-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}phenyl)-6-(piperidin-4-yl)-3,4-dihydropyrimidin-4-one
N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[2-(1H-pyrazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
2-amino-7-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
(3R,4R)-1-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
1-[4-(furan-2-yl)phenyl]-N-[3-(1H-imidazol-1-yl)propyl]piperidin-4-amine
N-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(pyrimidin-2-yl)piperidin-3-amine
2-{1-benzyl-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[3-(methylsulfanyl)propyl]-3-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
(3S,9aR)-3-(cyclohexylmethyl)-8-[4-(trifluoromethyl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-2-amine