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N-[(3R,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]pyridine-3-carboxamide
N-{3-[(pyridin-3-yl)amino]propyl}-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
5-{[(2-methyl-1H-indol-5-yl)methyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[2-(diethylamino)ethyl]-N-ethyl-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-({1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperidin-4-yl}methyl)benzoic acid
2-(2,5-dioxoimidazolidin-1-yl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]acetamide
4-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}benzoic acid
diethyl({[2-ethyl-5-(3-propoxypiperidine-1-carbonyl)furan-3-yl]methyl})amine
N-cyclopropyl-N-(naphthalen-1-ylmethyl)-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]acetamide
1-(2-methanesulfonylethyl)-4-{[3-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazine
2-methyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenol
N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]-3-[(2-fluorophenyl)formamido]propanamide
1-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(propan-2-yloxy)ethan-1-one
N-(1-methylpiperidin-4-yl)-7-oxo-N-(pyridin-4-ylmethyl)-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
1-[1-(furan-3-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
4-{[6-(dimethylamino)pyridin-3-yl]methyl}-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
1-[2-(1-cyclopropanecarbonylpiperidin-2-yl)ethyl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
2-(3-methylbut-2-en-1-yl)-8-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2,8-diazaspiro[4.5]decan-3-one
6-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-5,6-dihydro-1,6-naphthyridin-5-one
5-methoxy-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-4-oxo-1,4-dihydropyridine-2-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-N-{[2-(trifluoromethyl)phenyl]methyl}propanamide
1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(methylamino)acetamide
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-phenoxypropanamide
2-chloro-N-[2-(piperidin-1-yl)ethyl]-5-(1H-pyrazol-1-yl)benzamide
N-(3-hydroxypropyl)-1-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
2-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperazin-1-yl}pyridine-3-carbonitrile
(1R,5R)-N,N-dimethyl-6-[(phenylcarbamoyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(1R,2S)-N-(propan-2-yl)-2-propyl-N-[(2,4,5-trimethoxyphenyl)methyl]cyclopropane-1-carboxamide
1-[2-({[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amino)-4-methylpyrimidin-5-yl]ethan-1-one
3-(4-hydroxyphenyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-1H-pyrazole-5-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(morpholine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-(3-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(carbamoylamino)-N-methyl-N-[(4-phenoxyphenyl)methyl]acetamide
2,3-dimethyl-N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1H-indole-7-carboxamide
N-[4-({[2-(4-hydroxyphenyl)ethyl]carbamoyl}methyl)phenyl]butanamide
4-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(5-{[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]methyl}pyrimidin-2-yl)benzenesulfonamide
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](ethyl)(2-phenylethyl)amine
4,4,4-trifluoro-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
3-(2-{4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}propyl)pyridine
(1S,5R)-3-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
dimethyl[2-(2-{1-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}-1H-imidazol-1-yl)ethyl]amine
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
5-(3-acetylphenoxymethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
(2S,4R)-4-cyclohexaneamido-N-ethyl-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]pyrrolidine-2-carboxamide
1-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}-N-(pyridin-2-ylmethyl)piperidin-4-amine
1-[3-(1H-pyrazol-1-yl)benzamido]-1,2,3,4-tetrahydronaphthalene-1-carboxylic acid
1-ethyl-4-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]piperidine