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N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(carbamoylmethyl)-N-methylpiperidine-4-carboxamide
1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1H-pyrazole-4-carboxamide
5-chloro-2-[4-(1-methylpiperidin-4-yl)piperidine-1-carbonyl]-2,3-dihydro-1H-indole
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-[(4-methylphenyl)amino]-2-phenylpropanamide
(2S,4S)-4-amino-1-{[2-(2-hydroxyethoxy)phenyl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(dimethyl-1,3-oxazole-4-carbonyl)-4-(4-methoxyphenoxy)piperidine
1-[(4-acetylphenyl)methyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
4-(4-{1-[3-(1,3-oxazol-5-yl)phenyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
5-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-3-(4-methoxyphenyl)-1H-pyrazole
2-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-3-yl]-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
1-cyclopentyl-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazin-2-one
1-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]urea
N-[(2R,4R,6S)-2-(4-chlorophenyl)-6-(6-methoxypyridin-3-yl)oxan-4-yl]acetamide
N-methyl-6-{[(3-methyl-1,2-oxazol-5-yl)methyl]amino}-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
N-[2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-N-methylmethanesulfonamide
1-ethyl-3-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-7-methyl-1,4-dihydro-1,8-naphthyridin-4-one
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidine
2-[3-(2-hydroxyethyl)-4-(1-methylpiperidin-4-yl)piperazin-1-yl]-4,6-dimethylpyridine-3-carbonitrile
1-{2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
1-[2-({[(3-fluorophenyl)methyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
4-(6-methylpyridazin-3-yl)-1-phenylpiperazin-2-one
4-[3-(2-phenylethyl)-1,2-oxazole-5-carbonyl]thiomorpholine
1-{1-[(2,3-difluoro-4-methylphenyl)methyl]piperidin-4-yl}-3-methylbutan-1-ol
1-{4-[1-butyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]thiophen-2-yl}ethan-1-one
3-[(3R,4S)-4-(dimethylamino)-1-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]piperidin-3-yl]propanoic acid
7-(2,2-dimethylhexanoyl)-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
5-ethyl-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,3-oxazole-4-carboxamide
N-{2-[4-(propan-2-yl)-1,3-thiazol-2-yl]ethyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N1-cycloheptyl-N2-(4-methylpyridin-2-yl)ethane-1,2-diamine
4-[5-(morpholin-4-ylmethyl)pyridin-2-yl]benzoic acid
1-{2-[ethyl(methyl)amino]propanoyl}-4-(2-methylphenoxy)piperidine-4-carboxylic acid
N-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
N-[1-(4-methanesulfonylphenyl)propyl]-1,4-dithiepan-6-amine
N-{1-[5-(ethylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]ethyl}-3,4-dimethoxybenzamide
2-cyano-N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)benzamide
1-(3-methyl-1,2-oxazole-5-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
methyl 2-[(3-methylpyridin-4-yl)methyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrrole-2-carbonyl)piperidine
4-[3,5-dimethyl-1-(1H-1,2,3,4-tetrazol-5-yl)-1H-pyrazol-4-yl]-N-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(4-methoxy-2-methylphenyl)-3-{1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}propanamide
N-(4-methoxy-2-methylphenyl)-2,7-diazaspiro[4.5]decane-2-carboxamide
(2S,4R)-4-amino-N-ethyl-1-({5-[(N-methylmethanesulfonamido)methyl]furan-2-yl}methyl)pyrrolidine-2-carboxamide
2-(4,6-dimethyl-1-benzofuran-3-yl)-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
ethyl 1-(2-oxo-2-phenylacetyl)-3-(2-phenoxyethyl)piperidine-3-carboxylate
4-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]benzonitrile
3-{[1-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)pyrrolidin-3-yl]methyl}benzamide
4-[4-(4-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
2-{2-[(dimethyl-1H-1,2,4-triazol-1-yl)methyl]propanamido}-N-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
1-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)benzoyl]-3-(1H-imidazol-2-yl)piperidine