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N5-benzyl-N6-(1-methoxypropan-2-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-{2-amino-4-[(cyclopropylmethyl)(methyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
6-{pyrazolo[1,5-a]pyridin-7-yl}-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-[(2-chloropyridin-3-yl)methyl]-8-fluoro-N-methylquinoline-2-carboxamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
4-[1-(4-methoxyphenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]azepane
1-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}azepane
1-{1-[(1-methyl-1H-indol-6-yl)methyl]piperidin-4-yl}piperidine-4-carboxylic acid
N-[(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)methyl]thiophene-2-carboxamide
1-[3-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)benzenesulfonyl]piperidin-4-ol
4-{[6-(hydroxymethyl)-1,4-oxazepan-4-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-(2-{[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]amino}ethyl)imidazolidin-2-one
N-{2-methoxy-4-[3-(3-methyl-1H-1,2,4-triazol-5-yl)propanamido]phenyl}butanamide
6-[(2-methylphenyl)methyl]-3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
5-(4-cyclohexylphenyl)-N-[3-(1H-imidazol-1-yl)propyl]-1,2,4-triazin-3-amine
(1S,5R)-3-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 5-{[2-(2-methoxyphenyl)-1H-imidazol-1-yl]methyl}furan-2-carboxylate
2-(5-fluoro-2-methylphenyl)-N-(furan-2-ylmethyl)-N-[2-(morpholin-4-yl)ethyl]acetamide
1-{3-[(2-methylpiperidin-1-yl)methyl]phenyl}-3-[2-(morpholin-4-yl)ethyl]urea
1-(1-cyclohexylpiperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
N-({1-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}methyl)-2-(4-methoxyphenyl)acetamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}acetamide
4-({[4-(dimethylamino)-5-fluoropyrimidin-2-yl]amino}methyl)benzene-1-sulfonamide
4-[4-(furan-3-carbonyl)-1,4-diazepane-1-carbonyl]-1,2-dihydroisoquinolin-1-one
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-2-oxo-1-oxaspiro[4.5]decane-4-carboxamide
8-(2,3-dihydro-1H-inden-2-yl)-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-({1-[(2-ethylpyrimidin-5-yl)methyl]pyrrolidin-3-yl}methyl)-3-(propan-2-yl)urea
[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]({[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
2-amino-6-(3,5-difluorophenyl)-4-(2,3-dimethoxyphenyl)pyridine-3-carbonitrile
1-[1-(4-fluorophenyl)-2,2-dimethylcyclopropaneamido]cyclopentane-1-carboxylic acid
1-benzyl-N,5-dimethyl-N-[1-(pyridin-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(3S,4R)-N,N-dimethyl-1-(5-phenyl-1,2,4-oxadiazol-3-yl)-4-propylpyrrolidin-3-amine
4-cyclopentyl-N-{3-[2-(dimethylcarbamoyl)ethyl]phenyl}-3-oxopiperazine-1-carboxamide
N,1,3-trimethyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
4-chloro-3-(2-{4-[(dimethylamino)methyl]phenyl}pyrrolidine-1-carbonyl)-1H-pyrazol-5-amine
3-[2-(3-methoxyphenoxy)ethyl]-N-(propan-2-yl)benzamide
1-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-3-(1-methyl-1H-1,2,3-benzotriazol-5-yl)urea
N-[(2-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)-4,5,6,7-tetrahydro-1,3-benzothiazole-2-carboxamide
2-amino-8-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-methyl-1'-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)-N-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-5-yl}acetamide
N-ethyl-2-methyl-N-[(5-methylfuran-2-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
N-[4-(benzyloxy)-3-chlorophenyl]-2-methyl-5-oxo-1,4-diazepane-1-carboxamide
diethyl({[2-ethyl-5-(1,2,3,6-tetrahydropyridine-1-carbonyl)furan-3-yl]methyl})amine
(4aR,8aS)-1-[2-(3-fluorophenyl)ethyl]-6-[(2,3,4-trimethoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
5,5-dimethyl-3-{2-[4-(3-methylphenoxy)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)but-3-enamide
7-({methyl[2-(oxan-2-yl)ethyl]amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
1-(furan-2-ylmethyl)-N-[1-(thiophen-3-yl)propan-2-yl]piperidine-4-carboxamide