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7-methoxy-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(3S,4R)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
3-(4-fluorophenoxymethyl)-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidine
2-[2-({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-5,6-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
9-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-[5-chloro-2-(prop-2-en-1-yloxy)phenyl]-1H-imidazole
1-(cyclopropylmethyl)-5-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-methoxy-3-{[4-(2-methoxyphenoxy)piperidin-1-yl]methyl}phenol
3-chloro-1-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
N-[2-(dimethylamino)ethyl]-5-(1H-pyrrole-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-[2-(5-chlorothiophen-2-yl)-1H-imidazol-1-yl]acetamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-benzothiophene-2-carboxamide
N-{[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-1-(pyrimidin-2-yl)piperidin-4-amine
N,2,3,5-tetramethyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(oxolan-3-ylmethyl)-4-(pyridin-2-ylmethyl)-1,4-diazepane
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
N-[(1-cyclohexylpiperidin-3-yl)methyl]-2-(2-oxo-1,3-oxazolidin-3-yl)-N-(pyridin-3-ylmethyl)acetamide
4-[1-(4-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]-1-methyl-1,4,9-triazaspiro[5.5]undecane
2-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzoic acid
N,N-diethyl-1-{[1-(2-oxo-2H-chromene-3-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
5-fluoro-2-[1-(1-methyl-1H-pyrrole-2-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
2-[4-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methoxy)phenyl]acetamide
5-({3-[2-(1-benzothiophen-3-yl)pyridin-4-yl]pyrrolidin-1-yl}methyl)pyrimidine
5-cyclopropanecarbonyl-1'-[(2-ethoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[2-(1-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
4-chloro-1,3-dimethyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
1-methyl-4-{[5-(2-propyl-1,3-thiazol-4-yl)-1,2,4-oxadiazol-3-yl]methyl}piperazine
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
3-[(3R,4S)-3-(3-ethoxypropanamido)-4-(propan-2-yl)pyrrolidin-1-yl]propanoic acid
3-[(3R,4S)-1-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-4-(dimethylamino)piperidin-3-yl]propan-1-ol
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-3-yl)ethan-1-one
2-ethyl-9-[(2-fluoro-5-methoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(4aS,7aR)-1-(5-methyl-1,3-oxazole-4-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
(1S,5R)-6-(1-methyl-1H-pyrazole-4-carbonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-(4-methoxyphenyl)-N-{[3-(methylsulfanyl)phenyl]methyl}acetamide
N,7-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N-cyclohexyl-3-{[4-(1H-imidazol-1-yl)phenyl]formamido}propanamide
3-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-ylmethyl]-N-[4-(propan-2-yl)-1,3-thiazol-2-yl]benzamide
1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-4-(thian-4-yl)piperazine
4-(methoxymethyl)-N,5-dimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,2-oxazole-3-carboxamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(pyridin-3-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-(4-ethenylphenyl)-3-methyl-1H-1,2,4-triazole
(1R,5R)-3-methanesulfonyl-6-{[3-(morpholin-4-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N,N-bis(2-methoxyethyl)-2,6-dimethylpyridine-4-carboxamide
(3aR,6aS)-2-methyl-5-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-octahydropyrrolo[3,4-c]pyrrole-1,3-dione