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(1S,5R)-3-(2-amino-5-methylpyrimidin-4-yl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
7-[(1-ethyl-1H-indazol-3-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
1-{6-hydroxy-4-[4-(pyrrolidin-1-yl)benzoyl]-1,4-diazepan-1-yl}ethan-1-one
(1R,5S,6S)-6-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-3-azabicyclo[3.1.0]hexane
(4aS,7aR)-1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-4-(cyclopropylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopropyl-N-({4-[3-(dimethylamino)propoxy]phenyl}methyl)-2-methylpropanamide
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]propanamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-(7-{[3-(methoxymethyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
2-{4-cyclopentyl-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-(2-hydroxyethyl)-N-(1-phenylethyl)-5-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl})methylamine
3-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-N-(3-methylphenyl)propanamide
N-(furan-2-ylmethyl)-N-(2-hydroxyethyl)-5-methyl-2-phenyl-1H-imidazole-4-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-methoxyacetamide
4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1,2,3-thiadiazole
5-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-4-methyl-2-(piperidin-1-yl)pyrimidine
(2S,4R)-4-amino-1-(6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-N-methylpyrrolidine-2-carboxamide
9-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(3-hydroxy-3-methylbutyl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]benzamide
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-[2-(methylsulfanyl)ethyl]piperidin-4-amine
5-propyl-1'-(quinolin-4-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
8-cyclopropanecarbonyl-2-[(1-ethyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(methylamino)-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)pyrimidine-5-carboxamide
2-cyclopropyl-8-{2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
9-(6-oxopiperazine-2-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4,4-difluoro-1-({5-[(4-methyl-1H-imidazol-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)piperidine
methyl[1-(3-methylpyridin-2-yl)propan-2-yl](1,3-thiazol-4-ylmethyl)amine
6-[(diethylamino)methyl]-N-[2-(thiophen-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
(1R,5S)-3-[(2-aminopyridin-3-yl)methyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
(4aS,8aR)-6-(6-methylpyridazin-3-yl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-(3-chloro-4-fluorophenyl)-3-{1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-4-yl}propanamide
8-(benzenesulfonyl)-2-benzyl-2,8-diazaspiro[4.5]decan-3-one
1-(cyclopropylmethyl)-4-(4-methanesulfonylphenyl)-1H-pyrazole
7-chloro-2-{[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
3-hydroxy-N-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
N-{[3-(2-chlorophenyl)-1,2-oxazol-5-yl]methyl}-2-methylimidazo[1,2-a]pyridine-6-carboxamide
4-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-1-methylpiperazin-2-one
(3R,4R)-4-amino-1-{[6-(dimethylamino)pyridin-3-yl]methyl}piperidin-3-ol
1-benzyl-5-(2-methyl-1,3-thiazol-4-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
3-({7-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine
6-ethyl-2-(1-ethyl-1H-pyrazol-4-yl)-N-methyl-N-propylquinoline-4-carboxamide
3-(1H-1,3-benzodiazol-1-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)propanamide
4-phenyl-N-[(1-propylpiperidin-3-yl)methyl]benzamide
2-{4-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]morpholin-3-yl}-N-phenylacetamide
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}amine
(4aR,7aS)-1-(2-methoxyethyl)-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[4-(1H-1,3-benzodiazol-1-yl)phenoxy]propanamide
8-(2-methoxyethyl)-9-oxo-N-[2-(thiophen-2-yl)ethyl]-2,8-diazaspiro[5.5]undecane-2-carboxamide
1-(2,2-diphenylethyl)-4-(pyridin-3-yl)piperidin-4-ol
(4aR,8aR)-2-cyclopentanecarbonyl-7-[(2,3-difluoro-4-methylphenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol