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5-(6-methyl-9H-purin-9-yl)pyridin-2-amine
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
N-{3-[({[5-(2-chlorophenyl)furan-2-yl]methyl}amino)methyl]-5-(4-methylpiperazine-1-carbonyl)phenyl}acetamide
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-ethyl-N-(2-methylprop-2-en-1-yl)-1H-pyrazole-4-carboxamide
5-(1-{[3,5-dichloro-4-(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidin-2-yl)-3-methyl-1,2,4-oxadiazole
(3aR,6aR)-2-cyclopentyl-5-(pyridin-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-benzyl{[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]amino}sulfonamide
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
(3S,4S)-1-(3-methoxypyrazin-2-yl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-{4-cyclopentyl-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
(1S,5R)-6-[2-(methylsulfanyl)benzoyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(4-fluoro-3-methylphenyl)-2-({[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)amino)acetic acid
4-{2-[1-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)piperidin-2-yl]ethyl}phenol
1-methyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}azepane-2-carboxamide
1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
2-{[4-(cyclohex-3-en-1-yl)-1H-1,2,3-triazol-1-yl]methyl}-4-methylpyridine
2-benzyl-9-(3,3,3-trifluoropropyl)-2,9-diazaspiro[5.5]undecan-3-one
(2R,6S)-4-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,6-dimethylmorpholine
N-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
2-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-2,7-diazaspiro[4.5]decane
2-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]pyridine-4-carbonitrile
[(1-cyclopentylpiperidin-4-yl)methyl]({[3-(ethoxymethyl)-4-methoxyphenyl]methyl})(oxolan-2-ylmethyl)amine
1-(2-methoxy-4-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
butyl 3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-4-(1H-indol-3-yl)butanamide
1-(1,3-benzothiazole-5-carbonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-{3-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidin-1-yl]-3-oxopropyl}-4-methylbenzamide
(2S,4S)-4-({[4-(benzyloxy)phenyl]methyl}amino)-1-(2,3-dihydro-1H-inden-2-yl)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
3-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-1-{2-[(3-methylpyridin-4-yl)amino]ethyl}urea
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-(2-propyl-1,3-thiazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
8-(5-ethoxy-2-methyl-1-benzofuran-3-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{4-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
[3-(hydroxymethyl)-1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl]methanol
(2S,4R)-4-amino-N,N-diethyl-1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}pyrrolidine-2-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[1-(pyrimidin-4-yl)ethyl]benzamide
4-{[3-(3-chlorophenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-methylpiperidine
2-butyl-5-chloro-4-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-1H-imidazole
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(furan-2-ylmethyl)piperidine-3-carboxamide
4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1-(4-methylphenyl)piperazin-2-one
3-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]urea
N-ethyl-2-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-4-carboxamide
6-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-5-chloropyridine-3-carboxylic acid
N-({6-[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]pyridin-3-yl}methyl)acetamide
2,7-dioxo-N-(4-phenylbutyl)-1,3-diazepane-4-carboxamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
4-ethyl-1-methyl-3-[1-(oxolan-3-ylmethyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(3-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}phenyl)methyl]morpholine
1-[(3R,4R)-4-cyclopropyl-4-hydroxy-3-methylpiperidin-1-yl]-3-[methyl(propan-2-yl)amino]propan-1-one
4-{3-[2-(3-fluorophenyl)piperidine-1-carbonyl]phenyl}morpholine
(3R,4S)-1-(2,3-difluoro-4-methoxybenzoyl)-4-propylpyrrolidin-3-amine