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4-({4-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperazin-1-yl}methyl)-1H-indole
2-amino-4-[3-(2-hydroxyethoxy)phenyl]-6-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
4-(benzyloxy)-1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
1-[1-benzyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-3-propylurea
3-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(methylsulfanyl)phenyl]urea
N-(1-benzothiophen-2-ylmethyl)-N-methyl-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
3-(2,5-dioxoimidazolidin-4-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]propanamide
({1-[(1-cycloheptanecarbonylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)urea
5-(hydroxymethyl)-2-methyl-4-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)pyridin-3-ol
[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl)[1-(pyridin-2-yl)ethyl]amine
4-(4-fluorophenyl)-1-[4-(pyrimidin-2-yl)piperazin-1-yl]butan-1-one
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
ethyl 3-[(4-fluorophenyl)methyl]-1-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)piperidine-3-carboxylate
2-(2-methoxy-4-{[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]methyl}phenoxy)acetamide
4-({3-[2-(1-benzofuran-2-yl)pyridin-4-yl]pyrrolidin-1-yl}methyl)-1H-pyrazole-3-carboxylic acid
N-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amine
2-(2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}phenyl)-1H-imidazole
5-(morpholine-4-sulfonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
(2S)-N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-[3-(1H-imidazol-2-yl)propyl]-3-(morpholine-4-carbonyl)benzene-1-sulfonamide
2-(2-fluoro-5-methoxyphenyl)-2-[methyl(1,2-oxazol-3-ylmethyl)amino]acetic acid
(2S)-2-acetamido-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(methylsulfanyl)butanamide
6-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
3-(2-hydroxyphenyl)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(quinolin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-(5-{[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}thiophen-2-yl)acetamide
3-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
2-(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazin-1-yl)-5-fluoro-N,N-dimethylpyrimidin-4-amine
N-[3-(2-ethoxyethoxy)phenyl]-4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carboxamide
N-[(4-ethylphenyl)methyl]-5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
1-[(5-chlorothiophen-2-yl)methyl]-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanamide
2-({1-[(4-ethylphenyl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methyl-N-[2-(methylamino)ethyl]acetamide
7-fluoro-3-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
1-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
ethyl 1-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamido)piperidine-3-carboxylate
2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-5-methylphenol
methyl (1R,3S,3aR,6aS)-3-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]-1,5-dimethyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-({3-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]phenyl}amino)acetic acid
2-(dimethylamino)-N-methyl-2-(4-methylphenyl)-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
1-(2-phenylethyl)-4-(pyrrolidin-3-yl)piperidine
6-({[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)-2-methylpyrimidin-4-ol
[(1-benzylpiperidin-4-yl)methyl](methyl){pyrazolo[1,5-a]pyrimidin-3-ylmethyl}amine
(3E)-1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pent-3-en-1-one
[(4-{[5-(methanesulfonylmethyl)pyridin-2-yl]oxy}phenyl)methyl]dimethylamine
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-3-butanamidobenzamide
N-[3-(pyridin-3-yl)phenyl]-4-(pyrrolidine-1-carbonyl)piperidine-1-carboxamide
2-({methyl[3-(oxolan-2-yl)propyl]amino}methyl)benzoic acid