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N-[2-(4-chlorophenyl)ethyl]-1-methyl-N-(pyridin-4-ylmethyl)piperidine-4-carboxamide
2-(4-methoxynaphthalen-1-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
6-ethyl-3-[2-(1H-pyrazol-1-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
[(3R,4R)-1-{6-[ethyl(methyl)amino]pyrimidin-4-yl}-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
3-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
(1S,5R)-6-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-cyclopentyl-N3-(3-methylbutyl)-4-oxo-N5-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
6-{2-[2-(4-methoxynaphthalen-1-yl)-1H-imidazol-1-yl]ethyl}pyrimidin-4-ol
3-(3-methyl-1H-pyrazol-1-yl)-N-{[6-methyl-2-(2-methylphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)propanamide
2-[2-(1-methylpiperidin-2-yl)ethyl]-1,2-dihydrophthalazin-1-one
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
3-[2-(2-cyclohexyl-1H-imidazol-1-yl)ethyl]pyridine
1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylamino)ethan-1-one
4-{3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}-3-methyl-1-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
[(2,3-difluoro-6-methoxyphenyl)methyl][(1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
1-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}ethan-1-one
[(3R,5R)-1-(2-fluoro-6-methoxybenzoyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
N-[(2-amino-1,3-thiazol-4-yl)methyl]-2-[(4-chlorophenyl)amino]acetamide
1-(4,6-dimethylpyrimidin-2-yl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidin-4-amine
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
3-[(propan-2-yl)sulfamoyl]-5-(pyrimidin-5-yl)benzoic acid
2-cyclohexanecarbonyl-7-[(2E)-hex-2-en-1-yl]-2,7-diazaspiro[4.5]decane
(3S,4S)-4-(3-methoxyphenyl)-1-[(3-methyl-1H-indol-2-yl)methyl]piperidin-3-ol
(1S,5R)-3-(3-fluoropyridin-2-yl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-benzyl-N,N-dimethyl-5-[(2-methylpropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{[2-(pyridin-3-yl)pyrimidin-5-yl]formamido}hexanamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}pyrimidin-2-amine
1'-(2-methyl-1H-pyrrole-3-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[(3-methoxyphenyl)methyl][(1-methyl-1H-1,3-benzodiazol-2-yl)methyl](prop-2-en-1-yl)amine
1-[4-(1,3-thiazolidine-3-carbonyl)phenyl]pyrrolidin-2-one
N-(2-methoxyethyl)-3-(piperidin-3-yl)-N-(thiophen-2-ylmethyl)benzamide
4-[2-(2-methylphenoxy)acetyl]-1-(4-methylphenyl)piperazin-2-one
2-cyclopropyl-9-(3-phenoxypropanoyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}benzonitrile
4-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[(1-{[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-3-ol
2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
(1-{1-[1-(4-fluoro-2-methylphenyl)piperidin-4-yl]piperidin-3-yl}piperidin-4-yl)methanol
2-(2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamido)-N-methylacetamide
2-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}benzoic acid
N-ethyl-5-methyl-N-[(5-methylfuran-2-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
2-{4-[3-(4-hydroxyphenyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
2-(4-chloro-2-methylphenoxy)-1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]ethan-1-one
(2S,4R)-1-(adamantan-2-yl)-N-[2-(4-fluorophenyl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
(3S,4S)-1-[(5-methylpyrazin-2-yl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
5-methyl-4-{[1-(pyrazin-2-yl)propan-2-yl]amino}thieno[2,3-d]pyrimidine-6-carboxylic acid
N-(1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}pyrrolidin-3-yl)acetamide
4-fluorophenyl (7S,9aR)-7-[(benzyloxy)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate