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N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,1,3-trimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(3S,4R)-4-(4-methylphenyl)-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidin-3-yl]acetamide
(1s,4s)-4-[1-(4-chlorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]cyclohexan-1-ol
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)oxolane-3-carboxamide
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}benzamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-3,5,7-trimethyl-1H-indole-2-carboxamide
(4aS,7aR)-1-(3-methylbut-2-en-1-yl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-1-(4-phenylpiperazin-1-yl)propan-1-one
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-(2-phenylpropyl)pyrrolidin-2-one
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)propanamide
6-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindole-2-carbonyl]-5-hydroxy-2-(4-methylphenyl)-2,3-dihydropyridazin-3-one
N,N,2-trimethyl-7-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(2-methyl-1,3-thiazol-4-yl)-1-{1-oxa-8-azaspiro[4.6]undecan-8-yl}ethan-1-one
1-{5-[({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)methyl]-1-methyl-1H-pyrrol-3-yl}ethan-1-one
2-methoxy-3-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
2-benzyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1,3-thiazole-4-carboxamide
2-[3-(4-fluorophenoxymethyl)piperidin-1-yl]pyrazine
benzyl 3-({[1-(methoxymethyl)cyclobutyl]formamido}methyl)piperidine-1-carboxylate
2-(3-methoxypropyl)-9-(5-methylpyrazine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
2-{4-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]morpholin-3-yl}-N-(oxan-4-yl)acetamide
2-amino-4-(furan-3-yl)-6-(3-methoxyphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(3aS,6aS)-2-ethyl-1-oxo-5-[4-(1H-pyrazol-4-yl)butanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(1-ethyl-1H-pyrazole-5-carbonyl)-3-(4-fluorophenoxymethyl)piperidine
(1S,5R)-3-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S,4R)-1-(1,3-benzothiazol-2-yl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
2-(ethylamino)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}pyrimidine-5-carboxamide
4-{2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carbonyl}-1,4-oxazepane
1-[3-(methylsulfanyl)propanoyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
1-[(4-fluorophenyl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-(2-chlorophenyl)-3-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}propanamide
6-({[2-(5-methylthiophen-2-yl)ethyl]amino}methyl)-1,4-oxazepan-6-ol
2-(5-{1-[(4,5-dimethylfuran-2-yl)methyl]pyrrolidin-2-yl}-1,2,4-oxadiazol-3-yl)pyridine
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-{2-methylthieno[3,2-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
3-(2-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-oxoethyl)imidazolidine-2,4-dione
butyl 2-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate
2-[methyl(piperidin-4-yl)amino]-1-(3-phenylpiperazin-1-yl)ethan-1-one
(3-{2-[1-(5-chloropyridin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-(2,3-dimethylphenyl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-[4-(2,2-dimethylpropyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-{[3-(3-methylbutyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}-2-(morpholin-3-yl)acetamide
7-[(3,4-difluorophenyl)methyl]-2-(4,4,4-trifluorobutyl)-2,7-diazaspiro[4.5]decane
2-(3-methoxyphenoxy)-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-[4-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
2-ethyl-5-{4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine-1-carbonyl}pyrimidine
2-(2-hydroxyethyl)-8-(4-methylpyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
(3S,4S)-1-{[4-(2-fluorophenyl)phenyl]methyl}piperidine-3,4-diol
1-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-4-phenylpiperazine
2-[5-(3,4-dihydro-2H-1-benzopyran-3-yl)-3-(3-fluorophenoxymethyl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-{[(2,5-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide