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1-(6-cyclopropylpyrimidin-4-yl)-4-(2-fluoro-5-methylphenoxy)piperidine-4-carboxylic acid
4-({4-methyl-5-[1-(4-methylpent-3-en-1-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-{8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-N-[(2-methoxyphenyl)methyl]acetamide
N-(4-{1-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1H-imidazol-2-yl}phenyl)acetamide
1-methyl-8-[(5-methyl-1H-imidazol-4-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-butoxy-1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
ethyl 1-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidine-4-carboxylate
(2S,4S)-4-amino-1-{[6-(dimethylamino)pyridin-3-yl]methyl}pyrrolidine-2-carboxylic acid
4-[4-phenyl-1-(pyrrolidin-3-yl)-1H-imidazol-5-yl]phenol
N-(2,5-dimethoxyphenyl)-3-(4-phenylpiperazin-1-yl)piperidine-1-carboxamide
N-[(5-methylpyrazin-2-yl)methyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
4-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
3-(4-fluorophenyl)-5-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-(2-hydroxyethyl)-1-{1-[(4-methoxynaphthalen-1-yl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
1-(2,6-dimethylpyridin-4-yl)-4-(3-phenyl-1H-pyrazole-4-carbonyl)piperazine
3-chloro-5-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}-2-acetamidoacetamide
2-(naphthalen-2-ylmethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
6-(2,3-dimethoxy-5-methylphenyl)-N-ethylpyridine-3-carboxamide
methyl 1-(2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,3-oxazole-4-carbonyl)piperidine-4-carboxylate
4-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
3-(2-oxo-2-{2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-yl}ethyl)imidazolidine-2,4-dione
methyl 3-(oxolane-3-amido)-1-(3-phenylpropyl)-5-{[1-(propan-2-yl)piperidin-4-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(2-{1-[2-(4-acetylphenoxy)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
(3S,4R)-1-[(8-chloroquinolin-2-yl)methyl]-3-ethyl-4-methylpiperidin-4-ol
[1-({methyl[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}methyl)cyclopropyl]methanol
[(2-ethylpyrimidin-5-yl)methyl](methyl)[(3-phenyl-1H-pyrazol-4-yl)methyl]amine
1-[(2,3-dimethoxyphenyl)methyl]-3-{[(furan-2-ylmethyl)(methyl)amino]methyl}-3-hydroxypiperidin-2-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N3-cyclopentyl-N3-(3-phenylprop-2-yn-1-yl)piperidine-1,3-dicarboxamide
N,N-bis(propan-2-yl)-2-{pyrazolo[1,5-a]pyrimidin-3-yl}benzamide
6-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
[(2-butyl-1H-imidazol-4-yl)methyl](methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
N-(2-methoxyethyl)-2-(pyridin-3-yl)-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-8-[4-(1H-pyrazol-1-yl)butan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(tert-butylsulfanyl)ethyl]-3-[(4-fluorophenyl)formamido]propanamide
1-{4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-3-phenylpropan-1-ol
1-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-1,2,3,4-tetrahydroquinolin-2-one
4-(hydroxymethyl)-1-(quinolin-8-ylmethyl)piperidin-4-ol
5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-2-(1H-pyrrol-2-yl)pyridine
2-(acetamidomethyl)-N-(quinolin-8-yl)-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
3-(5-methylfuran-2-yl)-N-[(1s,4s)-4-aminocyclohexyl]benzamide
N-{2-methoxy-5-[2-(5-oxopyrrolidin-2-yl)acetamido]phenyl}furan-2-carboxamide
N4,5-dimethyl-N4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]pyrimidine-2,4-diamine
N-(1-cyclopentyl-1H-pyrazol-5-yl)-3-(thiophene-2-carbonyl)piperidine-1-carboxamide
1-methyl-4-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}piperazin-2-one
2-{[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]methyl}pyridine
2-{[(2S)-2-carbamoylpyrrolidin-1-yl]methyl}-4-hydroxyquinoline-6-carboxamide
N-benzyl-4-(ethylamino)-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
N-cyclopentyl-N-({4-[(3-fluorophenyl)methoxy]-3,5-dimethoxyphenyl}methyl)thiophene-2-sulfonamide