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8-(cyclohex-3-ene-1-carbonyl)-2-[(3,4-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-cyclopentyl-N3-(3-methylbutyl)-4-oxo-N5-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[4-chloro-3-(methylcarbamoyl)phenyl]-4-cyclopentyl-3-oxopiperazine-1-carboxamide
({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]amine
4,6-dimethyl-3-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-1,2-dihydropyridin-2-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}propanamide
4-methyl-1-{2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,3-triazole
N-{2-[4-(dimethylamino)phenyl]ethyl}-2,2-dimethyloxane-4-carboxamide
4-(5-fluoropyridine-2-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(1-phenyl-1H-pyrazol-5-yl)-1-(thiolan-3-yl)-1H-imidazole
2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]pyridine-4-carboxamide
N3-(1H-1,3-benzodiazol-2-ylmethyl)-N5-ethyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][(1-methyl-3-phenyl-1H-pyrazol-5-yl)methyl]amine
[5-({[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl)amino}methyl)-2-ethoxyphenyl]methanol
1-[4-({3-[(3S)-3-hydroxypyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)-3-methoxyphenyl]ethan-1-one
3-[(3R,4S)-1-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
N-benzyl-N-methyl-1-(pyridin-3-ylmethyl)piperidin-3-amine
N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
1-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
1-(2-{methyl[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]amino}ethyl)piperidin-2-one
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-cyclohexyl-8-methoxy-N-(pyridin-4-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-({1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-3-yl}methyl)-2-(2-methoxyphenoxy)acetamide
1-(1-benzoxepine-4-carbonyl)-4-(hydroxymethyl)piperidin-4-ol
5-(1-butylpyrrolidin-2-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}thiophene-2-carboxamide
2-{[(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amino]methyl}pyridine-3-carboxylic acid
1-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-2-(morpholin-2-yl)ethan-1-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}benzamide
N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-(pyridin-2-yl)piperidine-1-carboxamide
N-(6-methyl-2H-1,3-benzodioxol-5-yl)-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
2-[4-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)piperidin-1-yl]acetamide
4-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]oxane-4-carbonitrile
1-(3,5-dimethylphenyl)-4-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperazin-2-one
3-(cyclobutylsulfamoyl)-N-methyl-N-(oxan-2-ylmethyl)benzamide
2-methoxy-3-[1-methyl-3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]pyridine
6-(2,3-dimethoxyphenyl)pyridine-3-carboxamide
2-oxo-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
1-[3-(4-fluorophenoxy)azetidin-1-yl]-2-hydroxy-3-(2-methylphenoxy)propan-1-one
2-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]pyridine-3-carbonitrile
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
N-[(2-methylphenyl)methyl]-2-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}acetamide
2-[(quinoxalin-2-ylmethyl)(thiophen-2-ylmethyl)amino]butan-1-ol
1-[2-benzyl-5-oxo-4-(2-phenylphenyl)piperazin-1-yl]butane-1,2-dione
(4aS,7aR)-1-(2-hydroxybenzoyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-(2-phenoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,4R)-1-(3,4-dichlorobenzoyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
2-[4-(3-methoxypyridin-2-yl)-1H-pyrazol-1-yl]-N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
N,4-dimethyl-N-[(4-phenoxyphenyl)methyl]-1H-pyrrole-2-carboxamide