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(2S)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)pyrrolidine-2-carboxamide
4-(2-methoxyphenyl)-2-methyl-1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)piperazine
N-[(3-fluorophenyl)methyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine
N-[(4-chlorophenyl)methyl]-2-(3-hydroxypropanoyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
(3S,4S)-1-(1,3-benzothiazol-2-yl)-4-cyclopropylpyrrolidine-3-carboxylic acid
N-{2-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-oxoethyl}methanesulfonamide
N-(3-chloro-4-methoxyphenyl)-3-[1-(propane-1-sulfonyl)piperidin-3-yl]propanamide
2-(4-chlorophenyl)-4-(5-propyl-1,2,4-oxadiazol-3-yl)morpholine
6-ethoxy-2-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)quinoline
N-[2-(3-methylthiophen-2-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
4-{[1-({2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)pyrrolidin-3-yl]methyl}benzoic acid
1-{2-[2-(4-fluorophenyl)azetidin-1-yl]-2-oxoethyl}azonan-2-one
{1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
(butan-2-yl)(1H-imidazol-2-ylmethyl)(3-phenylprop-2-yn-1-yl)amine
5-(morpholin-4-ylmethyl)-N-{2-[(pyridin-3-yl)amino]ethyl}furan-3-carboxamide
[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
2-(furan-2-yl)-5-{5-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyrimidine
(2S,4R)-4-(dimethylamino)-1-{2-methyl-3-[(pyridin-2-ylmethyl)amino]benzoyl}pyrrolidine-2-carboxylic acid
1-methyl-4-(3-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-pyrazol-3-yl}phenyl)-1H-pyrazole
3-[(2R,3R,6R)-5-(3,5-difluoropyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
4-{1-[2-(4-ethylpiperazin-1-yl)acetyl]piperidin-3-yl}benzoic acid
4-{[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]sulfonyl}-N-methylbenzamide
2-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]pyridine-3-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(1H-pyrrol-2-yl)pyridine-3-carboxamide
4-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-(2-phenylethyl)piperazin-2-one
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-3-(pyridin-3-yl)propanamide
(1S,5R)-3-benzyl-6-[(1-propyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-{1-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
1-methyl-4-phenyl-3-{[1-(propane-2-sulfonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(3,5-dimethylphenyl)-4-(3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)piperazin-2-one
3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(piperidin-4-yl)piperidine
N-[1-(morpholine-4-carbonyl)azepan-3-yl]methanesulfonamide
2-methoxy-N,N-bis(propan-2-yl)-6-[6-(1H-pyrazol-1-yl)pyrimidin-4-yl]benzamide
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
N-(3-hydroxypropyl)-1-(3-propyl-1H-pyrazole-5-carbonyl)piperidine-3-carboxamide
1-[2-(1H-imidazol-5-yl)ethyl]-3-phenyl-5-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepin-9-yl}-1H-1,2,4-triazole
N-(2,3-dihydro-1H-inden-2-yl)-2-(2,5-dioxoimidazolidin-4-yl)-N-methylacetamide
1-{6-chloro-3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-3-(1-methyl-1H-imidazol-2-yl)piperidine
6-(2,5-dimethylfuran-3-yl)-7-methyl-N-(oxan-3-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-(4-methylpyrimidin-2-yl)-2-(piperidin-1-ylmethyl)-1,4-oxazepane
3-[2-methoxy-2-(thiophen-2-yl)ethyl]-3H,4H-pyrido[4,3-d]pyrimidin-4-one
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
benzyl (1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-{5-[2-(3-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}acetamide
N-[2-(2-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-[(3-methoxyphenyl)methyl]-N-(2-methylpropyl)acetamide
7-fluoro-2-methyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}quinoline-4-carboxamide
N-[2-(cyclohexylsulfanyl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(3,5-dimethoxyphenyl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine