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1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-(pyridin-4-yl)ethan-1-one
N-(butan-2-yl)-5-chloro-4,6-dimethyl-2-oxo-N-(thiophen-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
(3S,7S,8aS)-7-{[(5-chlorothiophen-2-yl)methyl]amino}-3-propyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3-methyl-4-oxo-N-[(1-propylpiperidin-3-yl)methyl]-3,4-dihydrophthalazine-1-carboxamide
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(pyrazin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3R,4R)-4-(hydroxymethyl)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-3-ol
3-[(cyclohex-1-en-1-ylmethyl)sulfamoyl]-N-(oxolan-3-yl)benzamide
1-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
4-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-2-ethoxyphenol
3-({[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)carbamoyl}amino)-4-chloro-N-methylbenzamide
5-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidine-1-carbonyl]-2-methylbenzene-1,3-diol
N-cyclopropyl-5-{1-[3-(furan-2-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-(3-{3-[(dimethylamino)methyl]-3-hydroxypiperidine-1-carbonyl}phenoxy)acetamide
ethyl 4-[(3-fluorophenyl)methyl]-1-(pyridine-3-carbonyl)piperidine-4-carboxylate
N-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-[benzyl({[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl})amino]ethan-1-ol
1-(3,5-dimethylphenyl)-4-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
1-[(2-butyl-1H-imidazol-4-yl)methyl]-N-(4-fluorophenyl)piperidin-3-amine
2-fluoro-6-[4-(hydroxymethyl)-4-methylpiperidine-1-carbonyl]phenol
2-[(dimethylcarbamoyl)amino]-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
(4aS,7aR)-1-[2-(4-methylphenyl)acetyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(dimethyl-1,3-thiazol-5-yl)-1H-1,3-benzodiazole-6-carboxylic acid
2-ethoxy-4-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
8-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]quinoline
3-(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-3-yl)-1-(4-methylpiperazin-1-yl)propan-1-one
1-(1-benzofuran-5-carbonyl)-2-methyl-4-(2-methylphenyl)piperazine
5-benzyl-N-[2-(1,3-thiazol-4-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(1S,5R)-3-[3-(4-fluorophenoxy)propyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
(3aR,6aR)-2-acetyl-5-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{[(3R,4S)-3-[2-(methylsulfanyl)acetamido]-4-(propan-2-yl)pyrrolidin-1-yl]methyl}benzamide
(1R,7S)-6-(2-phenylpyrrolidine-1-carbonyl)-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
[(3R,4S)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[(6-methylquinolin-5-yl)methyl]pyrrolidin-3-yl]methanol
1-(3-fluorophenyl)-3-(1-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
methyl 1-[(4-methyl-1,3-thiazol-5-yl)methyl]-3-(2-methylpropyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
2-[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-N-(4-methoxyphenyl)acetamide
(butan-2-yl)[(2-methoxypyrimidin-5-yl)methyl](pyridin-4-ylmethyl)amine
4-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
4-(1H-imidazol-1-ylmethyl)-1-[(6-methylpyridin-2-yl)methyl]piperidin-4-ol
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2,4-dimethoxybenzamide
3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[phenyl(pyridin-4-yl)methyl]propanamide
N3-benzyl-N3-methyl-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-2-(3,4-dichlorophenyl)morpholine
(4S,4aS,8aS)-4-phenyl-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-decahydroquinolin-4-ol
1-[7-(1-benzothiophen-3-yl)-9-ethoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
(3R,4S)-1-[4-(2-methylphenyl)benzoyl]-4-propylpyrrolidin-3-amine
2-(2,3-dihydro-1H-inden-1-yl)-N-(2-methoxyethyl)-N-(pyridin-2-ylmethyl)acetamide
methyl 5-[4-(3-methoxyphenyl)-3-methyl-5-oxopiperazin-1-yl]-5-oxopentanoate
3,3-dimethyl-1-[(3S,4R)-1-(1-methyl-1H-indole-4-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]urea
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide