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3-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-N-(2-methyl-1,3-benzothiazol-6-yl)piperidine-1-carboxamide
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(4,6-dimethylpyrimidin-2-yl)methyl]amine
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(2-methoxyacetyl)pyrrolidin-3-yl]pyrazine-2-carboxamide
3-(2,5-difluorobenzoyl)-1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidine
2-{2-[3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-2-oxoethyl}-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
8-(2,3,4,9-tetrahydro-1H-carbazole-7-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
2-{[(8-hydroxyquinolin-2-yl)methyl](methyl)amino}-N,N-dimethylpropanamide
methyl[(1-phenyl-1H-pyrazol-4-yl)methyl][(1-phenyl-1H-pyrazol-5-yl)methyl]amine
4-cyano-N-[(3R,4S)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]oxane-4-carboxamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]oxane-4-carboxamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
1-(4-ethoxy-3-methylphenyl)-4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}butane-1,4-dione
[(2S,6S)-4-(5-fluoro-1,3-dimethyl-1H-indole-2-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
1-benzyl-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]piperidin-4-amine
(3R,4S)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
8-{3-methyl-5-[(pyrimidin-2-ylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl}quinoline
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-methyl-N-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}acetamide
(3S,4S)-4-(4-fluorophenyl)-1-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
(3S,4R)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]benzamide
N-[3-(4-fluorophenyl)phenyl]-1-[2-(pyridin-3-yl)acetyl]piperidine-3-carboxamide
6-[3-(2-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-9H-purin-2-amine
4-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
4-(pyrazin-2-yl)-N-{3-[(trifluoromethyl)sulfanyl]phenyl}piperazine-1-carboxamide
1-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]-4-(3-methylpyridin-2-yl)piperazine
benzyl({[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl})(cyclopropylmethyl)amine
2-[3-(2-phenylethyl)piperidine-1-carbonyl]-4-(1H-1,2,3,4-tetrazol-1-yl)phenol
methyl (2S)-1-{2-[4-(4-{[(5-chlorothiophen-2-yl)methyl]amino}piperidin-1-yl)phenyl]acetyl}pyrrolidine-2-carboxylate
2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-4-(propan-2-yl)-1,3-thiazole
2-(ethylamino)-N,4-dimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-thiazole-5-carboxamide
3-{5-[4-(pyrrolidin-1-yl)benzoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
3-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide
7-(cyclopropylmethyl)-2-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-[1-(oxolan-3-ylmethyl)-1H-imidazol-2-yl]pyridine
{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
N-butyl-N-[(2-fluorophenyl)methyl]-2-(1H-pyrazol-1-yl)acetamide
8-[2-(naphthalen-1-yl)ethanesulfonyl]-2,8-diazaspiro[4.5]decan-3-one
N-ethyl-6-[3-(1-methoxyethyl)phenyl]pyridazin-3-amine
3-[2-(dimethylamino)ethyl]-8-(1H-indol-2-ylmethyl)-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-chloro-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-6-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}acetamide
N-[(2,3-dimethoxyphenyl)methyl]-2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)thiophene-2-sulfonamide
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[methyl(pyridin-2-ylmethyl)amino]acetic acid
3-(2-amino-4-methyl-6-{[2-(2-oxoimidazolidin-1-yl)ethyl]amino}pyrimidin-5-yl)propanoic acid
N-[1-(3-phenylpropyl)piperidin-3-yl]-4-(1H-1,2,4-triazol-1-yl)butanamide
(1R,2S)-N1-butyl-N2-(1H-indol-2-ylmethyl)cyclohexane-1,2-dicarboxamide