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(2S,4S)-4-amino-1-(2-methyl-4-phenyl-1,3-thiazole-5-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
5-(4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)-1-azabicyclo[3.2.1]octane
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
8-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
N-[2-(1H-imidazol-4-yl)ethyl]-3-(piperidin-3-yl)benzamide
8-{3-methyl-5-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-1,2,4-triazol-1-yl}quinoline
2-methoxy-5-({[(2-methoxyphenyl)methyl](propyl)amino}methyl)benzoic acid
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-methyl-6H,7H-pyrazolo[1,5-d][1,2,4]triazin-7-one
(1S,5R)-N-(3-methylphenyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
4-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-6-(4-methyl-1H-pyrazol-1-yl)pyrimidine
3-fluoro-4-methyl-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]benzamide
1-(2-{6-hydroxy-4-[(2-methylphenyl)methyl]-1,4-diazepan-1-yl}-2-oxoethyl)pyrrolidin-2-one
4-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propanoyl]-1-phenylpiperazin-2-one
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-[3-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methanol
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]propanamide
ethyl 4-benzyl-1-(pyridin-2-ylmethyl)piperidine-4-carboxylate
2-(methylsulfanyl)-1-{4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}ethan-1-one
N-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-6-methyl-4-(4-methyl-1H-imidazol-5-yl)-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
4-[5-(3-ethyl-5-methyl-1,2-oxazol-4-yl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
1-(1H-indazol-6-yl)-4-(4-oxo-4-phenylbutyl)piperazin-2-one
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-3-(pyridin-4-yl)propanamide
1-(2-oxo-2-{spiro[azepane-4,2'-chromene]-1-yl}ethyl)pyrrolidin-2-one
(4aS,8aR)-1-(2-aminoethyl)-6-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-decahydro-1,6-naphthyridin-2-one
3-[4-(2-ethylpyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]-N-(1,3-thiazol-2-yl)propanamide
4-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carbonyl]-1λ6-thiane-1,1-dione
5-({[(3-{2-[4-(4-methoxybenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]benzamide
4-(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
2-methyl-6-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)pyrimidin-4-ol
2-[3-({3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)phenyl]pyridine
N-(furan-2-ylmethyl)-4,6-dimethyl-2-oxo-N-(thiophen-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
3-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-oxoethyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
6-ethyl-1,5-dimethyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[5-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-carbonyl)thiophen-2-yl]ethan-1-one
1-[(1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
1-{4-[4-(4-aminopiperidin-1-yl)piperidin-1-yl]phenyl}pyrrolidin-2-one
(3aS,6aS)-2-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-5-pentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(3-chloro-4-propanamidophenyl)-2-(pyridin-2-ylsulfanyl)propanamide
1-{2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-oxoethyl}-3-methyl-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(4-phenyl-1-{3-[(pyridin-3-yl)amino]propyl}-1H-imidazol-5-yl)phenol
1-[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]-2-methoxy-2-methylpropan-1-one
3-{[3-(naphthalene-2-carbonyl)piperidin-1-yl]sulfonyl}pyridine
1-(2H-1,3-benzodioxol-5-ylmethyl)-5-(1,4-dioxan-2-yl)-1H-1,2,4-triazole
5-amino-2-ethyl-1-(3-methoxypropyl)-N-[(5-methylfuran-2-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
4-[2-(5-chloro-2-methoxypyridin-4-yl)-5-fluoropyrimidin-4-yl]morpholine
cyclopentyl 4-(4H-1,2,4-triazol-4-yl)benzoate
2-{4-[4-(1-phenylethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}acetic acid
N-(3-cyano-4-ethoxyphenyl)-4-(1H-pyrrole-2-carbonyl)piperazine-1-carboxamide