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N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-[3-(pyridin-3-yl)propyl]piperidine-3-carboxamide
4-(2-methylphenoxy)-1-(oxane-2-carbonyl)piperidine-4-carboxylic acid
[1-(6-aminopyrimidin-4-yl)-4-[(4-methoxyphenyl)methyl]piperidin-4-yl]methanol
N-cyclopropyl-3-{5-[(2-methoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-(1,3-diethyl-6-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-2-(morpholin-3-yl)acetamide
1-[3-(prop-2-en-1-yloxy)phenyl]-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
ethyl 4-{pyrazolo[1,5-a]pyrimidine-2-amido}piperidine-1-carboxylate
1-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-4-methylpiperazine
N-(furan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
(3R,5S)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
5-({[3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amino}methyl)-N-(propan-2-yl)pyrimidin-2-amine
5-(hydroxymethyl)-2-methyl-4-({methyl[1-(pyridin-3-yl)propyl]amino}methyl)pyridin-3-ol
9-[2-(2-methylphenyl)acetyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-4-(3-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}phenyl)butan-2-ol
8-methoxy-5-[6-(2-methoxyphenyl)pyridazin-3-yl]-2-methylquinoline
4-[(1R)-1-(4-fluorophenyl)ethyl]-3-(4-hydroxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
methyl 2-(pyrrolidine-1-sulfonyl)-6-(4,4,4-trifluorobutyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(2R,3R,6R)-5-cyclopropanecarbonyl-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(5S,9aS,9bS)-2-methyl-5-[4-(1H-pyrazol-1-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-butyl-2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(pyridin-3-yl)propan-1-one
1-cyclopentyl-4-[4-(piperidin-3-yl)benzoyl]piperazin-2-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(phenylsulfanyl)acetamide
3-[(4-cyanopiperidin-1-yl)sulfonyl]-N-(1-methyl-6-oxopiperidin-3-yl)benzamide
N-(1-methyl-1H-indazol-3-yl)-2-(1H-1,2,4-triazol-1-yl)acetamide
4-{4-[2-(2-chlorophenyl)acetyl]-5-methyl-2-oxopiperazin-1-yl}benzonitrile
1-{[3-fluoro-2-(trifluoromethyl)phenyl]methyl}-3-methylimidazolidin-2-one
1-{[(3S,4S)-3-hydroxy-1-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidin-4-yl]methyl}-3,3-dimethylurea
N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]acetamide
N-(2-methoxybutyl)-2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetamide
5-(4-ethoxyphenyl)pyrimidine
1-methyl-3-[2-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
8-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N2,N2-dimethyl-N5-{[4-(propan-2-yloxy)phenyl]methyl}-5,6,7,8-tetrahydroquinazoline-2,5-diamine
9-ethyl-1-methyl-4-(4,4,4-trifluorobutanoyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[1-(methoxymethyl)cyclobutanecarbonyl]-1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-propoxypiperidine
2-(methylamino)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,3-thiazole-4-carboxamide
7-methoxy-5-(1,2,3,4-tetrahydroisoquinolin-5-yl)-1-benzofuran-2-carboxylic acid
5-cyano-4-methyl-N-(1-methylpiperidin-4-yl)-6-oxo-N-(2-phenylethyl)-1,6-dihydropyridine-3-carboxamide
(4aR,7aS)-1-(2-methoxyethyl)-4-(quinoline-6-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
2-(cyclohex-1-en-1-yl)-N-{[2-(2-acetamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}acetamide
3-{[(2,2-dimethyloxan-4-yl)(methyl)amino]methyl}-N-(1-ethyl-1H-1,2,4-triazol-5-yl)benzamide
N-[2-(dimethylamino)-2-(thiophen-2-yl)ethyl]-2-(1H-imidazol-2-yl)benzamide
4-(3-hydroxypropanoyl)-1-(3-methoxyphenyl)piperazin-2-one
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N,1-dimethyl-N-[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrrolidine-3-carboxamide
2-tert-butyl-N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-4-hydroxy-N-methylpyrimidine-5-carboxamide