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2-cyclopropyl-N-[2-(4-ethoxyphenyl)ethyl]pyrimidine-5-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-4-(1H-pyrazol-1-yl)benzamide
6-[(diethylamino)methyl]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-tert-butyl-N-{[5-(methoxymethyl)furan-2-yl]methyl}-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-amine
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-4-methyl-1H-imidazole-2-carboxamide
(4aS,7aR)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(1H-imidazol-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N,N-dimethyl-3-(3-phenylphenyl)-1H-1,2,4-triazol-5-amine
butyl 9-oxo-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecane-2-carboxylate
8-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)imidazo[2,1-b][1,3]thiazole-5-carboxamide
1-[2-(3-benzyl-1H-1,2,4-triazol-5-yl)ethyl]-4-(3-methylphenyl)piperazine
(4aS,8aR)-1-(2-aminoethyl)-6-[1-(4-fluorophenyl)cyclopropanecarbonyl]-decahydro-1,6-naphthyridin-2-one
(2S,4S)-N-ethyl-4-(2-hydroxybenzamido)-1-[(5-methylfuran-2-yl)methyl]pyrrolidine-2-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,2,6-trimethylquinoline-4-carboxamide
N-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl}-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-(1H-indol-3-yl)-N-{1-oxa-8-azaspiro[4.5]decan-3-yl}propanamide
8-methoxy-5-[6-(1H-pyrazol-1-yl)pyrimidin-4-yl]quinoline
2-(5-{2-oxa-7-azaspiro[4.5]decane-7-carbonyl}-1H-1,3-benzodiazol-1-yl)ethan-1-ol
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-{[2-(1,3-thiazol-4-yl)acetamido]methyl}benzoate
N-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-[2-ethyl-4-(pyridin-4-yl)phenyl]acetamide
ethyl 1-(6-methylquinoline-4-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
2-{[3-(5-chloro-2-methoxybenzoyl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
(1R,5R)-6-[(5-acetylthiophen-3-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
(4aS,8aR)-6-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
11-benzoyl-4-[(1-ethyl-1H-imidazol-2-yl)methyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
N5-benzyl-N3-methyl-4-oxo-1-(propan-2-yl)-N3-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(pyridine-3-sulfonyl)-decahydro-1,6-naphthyridin-2-one
N-{1-[4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carbonyl]piperidin-4-yl}methanesulfonamide
2-methyl-4-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-5-propylpyrimidine
3-methyl-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}furan-2-carboxamide
2-[({1-[3-(piperidin-3-yl)benzoyl]piperidin-4-yl}oxy)methyl]pyridine
2-(ethylamino)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrimidine-5-carboxamide
N-(1-{1-[(3-chloro-4-hydroxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
4-(6-methylpyridine-3-carbonyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(1-ethyl-1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{4-[(2,3-dihydro-1H-inden-1-yl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
4-(4-acetylphenyl)-2-methoxypyridine-3-carbonitrile
2-[(3-fluorophenyl)methyl]-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}morpholine
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
1-(4-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methoxy}phenyl)propan-1-one
N-cyclohexyl-N-({1-[(2S)-2,3-dihydroxypropyl]-1,2,3,6-tetrahydropyridin-4-yl}methyl)acetamide
1-benzoyl-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methylpiperidin-4-amine
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2,3-dihydro-1H-inden-2-amine
N-[2-(azepan-1-yl)-2-phenylethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-{[(2S,4S)-4-fluoro-1-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)pyrrolidin-2-yl]methyl}methanesulfonamide
N-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]pyrimidin-2-amine