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2-{5-[(dimethyl-1,3-thiazol-5-yl)methyl]-1-(2-hydroxybutyl)-1H-1,2,4-triazol-3-yl}acetamide
7-(1H-imidazol-4-ylmethyl)-N-(2-phenylethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(2-phenoxypyridin-3-yl)methyl]pyridine-4-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-3-(pyridin-2-yl)propan-1-one
5-methyl-1'-(5-phenyl-1,2-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(1S,5R)-6-(2-ethoxyethyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-{2-methyl-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-2-yl}morpholine
2-{[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]amino}propane-1,3-diol
N-[3-(furan-2-yl)propyl]thiolan-3-amine
1-[4-(hydroxymethyl)benzoyl]-4-(3-methoxypropyl)-1,4-diazepan-6-ol
(2R,6S)-4-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-2,6-dimethylmorpholine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,3-dimethyl-1H-pyrazole-4-carboxamide
2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
2-{[5-(3-methylthiophen-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}pyridine
N-[3-(4-methylpiperazin-1-yl)propyl]quinoxaline-5-carboxamide
3-[(2,4-difluorophenyl)methyl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-3-carboxylic acid
3-[5-(5-methyl-1,3-oxazol-4-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]pyridine
2-(2-{1-[4-(piperidin-1-yl)benzoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
4-{[5-(2,5-dimethoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]methyl}pyridine
2-{8-[2-(methylsulfanyl)benzoyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetic acid
(1S,5R)-6-(4-methyl-1H-imidazole-2-carbonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-[(3-methylpyridin-4-yl)methyl]-1,3-oxazole-4-carboxamide
3-cyclopropyl-N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-1H-pyrazole-5-carboxamide
2-[(adamantan-1-ylmethyl)(5-phenyl-1,2,4-triazin-3-yl)amino]ethan-1-ol
2-cyclobutyl-1-methyl-7-(oxolane-2-amido)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
N-[(3S,4R)-1-(1H-imidazol-2-ylmethyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
6-[4-(5-propyl-1,2-oxazole-3-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
N-[2-(dimethylamino)-2-(pyridin-2-yl)ethyl]-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-({1-[2-(carbamoylamino)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}methyl)cyclohexanecarboxamide
3-[3-(ethoxymethyl)-1-ethyl-1H-1,2,4-triazol-5-yl]-N,N-dimethylpropanamide
3-(1H-1,3-benzodiazol-1-yl)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]propanamide
N-(1-cyclopropanecarbonylpiperidin-3-yl)-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
(2S)-2-({5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazol-3-yl}formamido)propanamide
N-(2-methoxyethyl)-1-[1-(6-oxo-1,6-dihydropyridine-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
7-(2-methoxyphenyl)-2-(2-methyl-1,3-thiazol-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]morpholine-2-carboxamide
(3S,4R)-1-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-4-methylpiperidine-3,4-diol
5-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
4-(5-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
N-ethyl-2-methyl-N-[2-(pyrrolidin-1-yl)ethyl]imidazo[1,2-a]pyrimidine-3-carboxamide
1-[2-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
3-({1-[(6-chloropyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
2-{2-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}benzamide
N-[(3-methoxyphenyl)methyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-methyl-5-phenyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1,2-oxazole-3-carboxamide
(2S,4R)-1-[(2,6-difluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-methyl-N-(1H-pyrazol-5-ylmethyl)pyrrolidine-2-carboxamide
1-ethyl-8-(furan-3-ylmethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-methyl-1-[2-(piperazin-1-yl)acetyl]-1,4-diazepan-5-one