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3-(4-chlorophenyl)-4-{[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}butanoic acid
(benzylsulfamoyl)[1-(4-methylpyridin-2-yl)propyl]amine
N'-[(1-butylpiperidin-4-yl)methyl]-N-cyclopentylbutanediamide
2-{10-oxo-3,9-diazaspiro[5.6]dodecane-3-carbonyl}benzonitrile
{[5-(1-cyclopentanecarbonylpiperidin-4-yl)-4-cyclopropyl-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
1-{[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
(3-{[ethyl(oxan-4-ylmethyl)amino]methyl}-2,4,6-trimethylphenyl)methanol
1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-4-(4H-1,2,4-triazol-3-ylmethyl)piperazine
1-{2-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-7-phenoxy-1,2,3,4-tetrahydroquinolin-2-one
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-{[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}piperidin-2-one
1-[2-(pyrrolidin-1-yl)butanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(4-acetylphenoxy)-N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)acetamide
1-(2,3-dihydro-1H-inden-2-yl)-4-(2-methyl-1,3-thiazole-5-carbonyl)-1,4-diazepane
3-(3-hydroxy-3-methylbutyl)-N-(thiolan-3-yl)benzamide
3-[1-(3-chlorobenzoyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
2-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-6-methoxyphenol
4-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-N,N-dimethyl-5,6,7,8-tetrahydroquinazolin-2-amine
2-[(2,3-dimethoxyphenyl)methyl]-4-[4-(5-methylthiophene-2-carbonyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-ethoxyethan-1-one
4-[5-({[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoic acid
(2S,4R)-4-amino-N-methyl-1-{[3-(morpholin-4-yl)phenyl]methyl}pyrrolidine-2-carboxamide
2-(3-{[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenyl)ethan-1-amine
2-(pyrimidin-2-ylsulfanyl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}ethan-1-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-[2-(3-fluorophenyl)ethyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-ethyl-5-[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-[1-benzyl-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-indole
1-phenyl-5-(2,4,5-trimethoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazole
1-(6-methyl-2-phenyl-1,2-diazinan-1-yl)-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
ethyl 3-[2-(2-chloro-4-hydroxyphenyl)-1H-imidazol-1-yl]propanoate
5-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)methyl]-3-(propan-2-yl)-1,2,4-oxadiazole
2-cyclopropyl-6-oxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,6-dihydropyrimidine-5-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}propan-1-one
2-{[3-(ethylsulfanyl)propanamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
(2S,4S)-4-amino-N-methyl-1-[2-(6-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)acetyl]pyrrolidine-2-carboxamide
(3S,9aR)-2,3-dimethyl-8-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(cyclohex-1-en-1-ylmethyl)-2-[4-(5-hydroxypyrazine-2-carbonyl)morpholin-3-yl]acetamide
3-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-4-yl}-1-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)quinoline
[(2-chloro-4-fluorophenyl)methyl][(1-ethyl-1H-pyrazol-4-yl)methyl]methylamine
1-[(5-ethylpyridin-2-yl)methyl]-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
N-(furan-3-ylmethyl)-N-methyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
2-[(2,3-dimethoxyphenyl)methyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(pentan-2-yl)-8-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[2-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]pyridine
2-chloro-4-{[(3,4-dihydro-2H-1-benzopyran-3-yl)amino]methyl}phenol
ethyl 2-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-6-methylpyrimidine-4-carboxylate
4-chloro-3-[1-(1,4-dioxan-2-ylmethyl)-1H-imidazol-2-yl]-1-methyl-1H-indazole
7-[2-(phenylamino)pyrimidine-5-carbonyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-{[1-(pyridin-3-ylmethyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide