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2-(3-{[(oxan-4-yl)carbamoyl]amino}phenyl)acetamide
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-4-(propan-2-yl)-1,3-thiazole-2-carboxamide
2-[3-(pyrrolidin-1-yl)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(methylsulfanyl)-5-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)pyrimidine
benzyl({[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})[(4-methyl-1,3-thiazol-5-yl)methyl]amine
(3S,4R)-1-(1H-imidazol-2-ylmethyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
8-{[2-(morpholine-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}quinoline
6,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-4-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}quinoline
3-{1-[(3-chloro-4-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-[5-(2-ethoxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(4-hydroxypiperidin-1-yl)propan-1-one
1-(2-methoxy-4-{[4-(pyrrolidin-1-yl)piperidin-1-yl]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
3-{5-[1-(quinolin-3-yl)-1H-imidazol-2-yl]thiophen-3-yl}prop-2-yn-1-ol
1-(pyrrolidin-1-yl)-3-[1-(thian-4-yl)piperidin-3-yl]propan-1-one
[(4-methanesulfonylphenyl)methyl](methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
5-[3-(1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-1H-pyrazol-3-yl)phenyl]pyrimidine
9-(2-fluoro-4-methylbenzoyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-4-({4-methyl-5-[1-(oxan-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperazine
3-(2-fluorophenoxymethyl)-N-(1H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
9-[2-(2,3-dimethylphenoxy)ethyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-5-{[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
(4aS,7aR)-1-[3-(1,3-benzothiazol-2-yl)propanoyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-5-methyl-N-(oxolan-2-ylmethyl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[(6-methylquinolin-5-yl)methyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethan-1-one
4-(2-{4-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)morpholine
(1R,3S)-1,3-dihydroxy-N-(2-phenylphenyl)-7-azaspiro[3.5]nonane-7-carboxamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propanamide
5-methoxy-2-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-4H-pyran-4-one
5-methyl-N-{4-[3-(2-oxooxolan-3-yl)propanamido]phenyl}furan-2-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperazine
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
3-(1-ethyl-1H-pyrazol-4-yl)-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(5-{[cyclopentyl(methyl)amino]methyl}-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl)acetic acid
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]acetamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]pyrrolidin-3-yl]methanol
N,6-dimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]imidazo[1,2-a]pyridine-2-carboxamide
1-(thian-4-yl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
{[2-(difluoromethoxy)phenyl]methyl}[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
5-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}-2-(pyridin-4-yl)pyrimidine
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(2,2-dimethyloxan-4-yl)-1H-pyrazole-4-carboxamide
1-(quinoxaline-5-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-2,3-dihydro-1-benzofuran-2-carboxamide
3-(1H-1,2,3-benzotriazol-1-yl)-1-{3-[4-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}propan-1-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}but-2-ynamide
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-phenoxypropan-1-one
4-(3-{4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}propyl)morpholine
N-{[1-(1,3-dihydroxypropan-2-yl)pyrrolidin-3-yl]methyl}-2-hydroxy-5-methylbenzamide
2-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-5-methoxy-4H-pyran-4-one