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1-amino-N-[3-(1H-indazol-1-yl)propyl]cyclopropane-1-carboxamide
3-[4-(3-methylphenyl)piperazin-1-yl]-N-[4-(1H-pyrazol-1-yl)butan-2-yl]propanamide
1-[6-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyridazin-3-yl]azepane
5-[(2-methoxyquinolin-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
2-[(2,3-dihydro-1H-inden-2-yl)amino]-N,N-bis(prop-2-en-1-yl)acetamide
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-(4-chlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-ethyl-6-[3-(2-methoxybenzoyl)piperidin-1-yl]pyridine-3-carboxamide
3-(3-chlorophenyl)-1-[3-(3-methoxypropyl)piperidin-1-yl]propan-1-one
1-(diethylamino)-3-[2-methoxy-5-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
{4-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]-1,4-oxazepan-6-yl}methanol
N-[(2S,4R,6S)-2-(4-chlorophenyl)-6-ethyloxan-4-yl]benzamide
4-{4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-1-yl}butan-1-ol
1-(2-ethoxyphenyl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}urea
2-{[3-(1H-pyrazol-1-yl)propyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-[(4-fluorophenyl)methyl]-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
4-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-4H-1,2,4-triazole
N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(piperidin-3-yl)benzamide
6-[3-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[1-(hydroxymethyl)cyclopentyl]methyl}-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(dimethylamino)-N-[3-({[2-(1-methylpyrrolidin-2-yl)ethyl]carbamoyl}amino)phenyl]acetamide
3-[5-(6-methoxy-3-methyl-1-benzofuran-2-yl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
N,N-dimethyl-2-[6-methyl-2-(morpholin-4-yl)pyrimidin-4-yl]aniline
(2S,4R)-4-{[(9-ethyl-9H-carbazol-3-yl)methyl]amino}-N-(2-methoxyethyl)-1-(propan-2-yl)pyrrolidine-2-carboxamide
2-(adamantan-1-yl)-N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-methyl-3-(morpholin-4-yl)propanamide
3-methoxy-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)propanamide
1-[(3-chlorophenyl)methyl]-4-(4-methyl-1,3-thiazole-5-carbonyl)piperazine
1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-phenylacetamide
3-cyclopropyl-5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-[(4-methylphenyl)methyl]-1H-1,2,4-triazole
N-(oxolan-2-ylmethyl)-7-(propan-2-yl)-N-(pyridin-2-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
4-[2-(3,4-dichlorophenyl)morpholin-4-yl]pyrimidin-2-amine
(2R,3R)-3-{[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-[1-(1,4-dimethyl-1H-indole-2-carbonyl)piperidin-4-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2-hydroxyethyl)-8-(2-methoxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
1-cyclopropyl-5-oxo-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}pyrrolidine-3-carboxamide
3-acetamido-N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}propanamide
1-{2-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
7-[1-(2-methylpropyl)-5-oxopyrrolidine-3-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
5-methyl-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-1H-indazole-3-carboxamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(quinoline-7-carbonyl)pyrrolidin-3-yl]methanol
(1S,5R)-6-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
6-(methoxymethyl)-2-{4-[(2-phenylazetidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
3-(4-chloro-1H-pyrazol-1-yl)-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
6-(3-carbamoylpiperidin-1-yl)-N-methyl-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
3-{[(1S,4S)-5-(3-chlorophenyl)-6-oxo-2,5-diazabicyclo[2.2.1]heptan-2-yl]methyl}-N-methyl-1,2,4-oxadiazole-5-carboxamide
2-[(2,4-dimethyl-1,4-diazepan-1-yl)methyl]-3,7-dimethyl-1H-indole
(2R)-2-[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-phenyl-1H-imidazol-1-yl]-3-hydroxypropanoic acid
(3aR,6aR)-2-(3-methylbut-2-en-1-yl)-5-(5-propylpyrimidin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid