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5-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-(furan-3-ylmethyl)-4-(2-methylquinolin-6-yl)piperidin-4-ol
7-(cyclopropylmethyl)-2-{[2-(trifluoromethyl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
7-(pyridin-2-ylmethyl)-4-(thiomorpholin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
6-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
6-oxo-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-1,4,5,6-tetrahydropyridazine-3-carboxamide
(2S,4R)-4-amino-1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
7-propyl-2-(1,2-thiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(3-methoxypropyl)-N-(2-phenylethyl)piperidine-1-carboxamide
2-[2-(3-chlorophenyl)acetyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
methyl 3-[({2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}carbamoyl)amino]benzoate
N-benzyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[(4-methyl-1,3-thiazol-5-yl)methyl]acetamide
7-(5,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-cyclopropyl-2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-{[4-(methylsulfanyl)phenyl]methyl}acetamide
3-(1H-1,2,3-benzotriazol-1-yl)-1-{9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}propan-1-one
5-methyl-1-(4-methylphenyl)-4-(1H-pyrrole-2-carbonyl)piperazin-2-one
(2R,6R)-4-acetyl-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-{4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]thiophen-2-yl}ethan-1-one
2-[(5-methylpyrazin-2-yl)methyl]-9-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-(5-methanesulfonyl-2-methylpyrimidin-4-yl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
4-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1S,5R)-6-methyl-3-{3-[5-(thiophen-2-yl)furan-2-yl]propanoyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(3,4-dimethylphenyl)-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-amine
2-methyl-4-[3-(3-propylmorpholine-4-carbonyl)phenyl]butan-2-ol
6-(1-benzothiophen-3-yl)-9H-purin-2-amine
2-methyl-1-{2-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,4-dihydroquinolin-4-one
(4aS,7aR)-1-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,4-dimethyl-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
2-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-N-(5-propyl-1,3,4-thiadiazol-2-yl)acetamide
3-(2-amino-1,3-thiazol-4-yl)-1-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]propan-1-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1H-pyrazole-4-carbonyl)piperazin-2-one
3-[4-(2-methanesulfonylethyl)piperazine-1-carbonyl]-2-methyl-1,2,3,4-tetrahydroisoquinoline
5-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
3-{2-oxo-2-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
2-amino-4-(1H-indol-5-yl)-6-(6-methoxypyridin-3-yl)pyridine-3-carbonitrile
4-[(3-{1-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-imidazol-2-yl}phenyl)methyl]morpholine
2-({[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-hydroxyethyl)amino)ethan-1-ol
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-(cyclohexylmethyl)-2-phenylacetamide
2-amino-4-[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
6-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
3-(oxolan-3-yl)-5-(3-propyl-1H-pyrazol-5-yl)-1,2,4-oxadiazole
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
N-ethyl-3-(3-fluorophenyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-pyrazole-4-carboxamide
6-{[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]methyl}-2-methylpyrimidin-4-ol
1-(furan-3-ylmethyl)-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
N-{[1-(2H-1,3-benzodioxol-5-ylmethyl)-4-hydroxyazepan-4-yl]methyl}piperidine-1-carboxamide
1-[(4-chlorophenyl)methyl]-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
(2S,4R)-N-ethyl-4-{imidazo[1,2-a]pyridine-3-amido}-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidine-2-carboxamide
2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyridine