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2-[(4-methoxy-4-methylpentan-2-yl)amino]-N,N-dimethylethane-1-sulfonamide
4-hydroxy-1-[6-(1-hydroxyethyl)pyridin-2-yl]piperidine-4-carboxylic acid
N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-{[(cyclopropylmethyl)amino]methyl}-1-[(2,3-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
6-[4-(2-phenoxyethyl)piperazine-1-carbonyl]quinoxaline
N-[1-(1H-imidazol-1-yl)butan-2-yl]-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-2-(5-oxopyrrolidin-2-yl)acetamide
N-(cyclobutylmethyl)-N-(oxolan-2-ylmethyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
9-(4-cyclopentylpyrimidin-2-yl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{2,7-diazaspiro[4.5]decane-7-carbonyl}-6-methoxy-1,4-dihydroquinolin-4-one
6-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-9H-purine
N,2-dimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]-3-[(pyridin-2-ylmethyl)amino]benzamide
5-[4-(aminomethyl)piperidin-1-yl]-2-({8-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2,3-dihydropyridazin-3-one
3,5-dimethyl-1-{1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}-1H-pyrazole
N-[2-methyl-1-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)propyl]-2-(trifluoromethyl)benzamide
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(naphthalen-1-yl)urea
3-[6-(hydroxymethyl)-1,4-oxazepane-4-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
5-{3-tert-butyl-1-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}thiophene-2-carboxylic acid
4-(hydroxymethyl)-N,N-dimethyl-4-(2-phenylethyl)piperidine-1-sulfonamide
N-(2,3-dihydro-1H-inden-2-yl)-1-(5-propylpyrimidin-4-yl)piperidin-4-amine
2,8-dimethyl-4-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoline
1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-(thiophen-3-yl)ethan-1-one
N-(3-methylphenyl)-3-[1-(pyrazine-2-carbonyl)piperidin-4-yl]propanamide
4-[3-(1-butyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)phenyl]-1λ6-thiomorpholine-1,1-dione
2-ethyl-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylpyrimidine-5-carboxamide
N-(2-methoxyethyl)-2-methyl-N-(pyridin-3-ylmethyl)-1-benzofuran-5-carboxamide
6-amino-N-({1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}methyl)pyridine-3-carboxamide
2-hydroxy-5-{[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]methyl}benzoic acid
2-{2-[1-(5-phenyl-1,3,4-thiadiazol-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
(3S)-4-[5-(1H-1,3-benzodiazol-1-ylmethyl)-1H-pyrazole-3-carbonyl]-1,3-dimethylpiperazin-2-one
3-[3-(3-ethyl-1,2,4-oxadiazol-5-yl)propyl]-1H-indole
5-[4-(4-acetylphenyl)piperazine-1-carbonyl]-1-(pyridin-2-ylmethyl)piperidin-2-one
2-{1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-3-carbonyl}pyridine
(1R,9S)-11-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
N-[1-(furan-2-carbonyl)piperidin-4-yl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-cyclopropyl-4-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
2-ethyl-9-(1-methyl-1H-imidazole-5-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
N-[3-(3-methylbenzamido)phenyl]-1,4-dioxane-2-carboxamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
4-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-4-oxobutane-1-sulfonamide
3-(2,3-dihydro-1H-inden-2-yl)-5-(2-phenylethyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
[3-({[3-(2-amino-1,3-thiazol-4-yl)propyl]amino}methyl)-2,4,6-trimethylphenyl]methyl acetate
3-cyclopropyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1H-pyrazole-5-carboxamide
(3S,4R)-4-(3-methylthiophen-2-yl)-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-ol
3-chloro-4-({1-[1-(4-hydroxyphenyl)propan-2-yl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}pyridine-3-sulfonamide
2-amino-4-(2-chlorophenyl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
[3-(cyclopropylmethyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidin-3-yl]methanol
2-amino-N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide