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8-(4-aminopyrimidin-2-yl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
(2S)-2,6-diamino-1-[4-(2-methylphenoxy)piperidin-1-yl]hexan-1-one
(3aR,6aR)-2-cyclopentyl-N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2,3-difluoro-6-methoxy-N-methyl-N-(1H-pyrazol-3-ylmethyl)benzamide
methyl 4-{[(2S,4R)-4-[(4-methoxyphenyl)sulfanyl]-2-(4-methyl-1,4-diazepane-1-carbonyl)pyrrolidin-1-yl]methyl}benzoate
4,6-dimethyl-1-{2-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
3-(1H-1,3-benzodiazol-1-yl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}propanamide
(3R,4R)-3-methyl-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(oxan-4-yl)piperidin-4-ol
N,N-dimethyl-3-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]propane-1-sulfonamide
1-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]piperidin-4-ol
1-(2-{3,9-diazaspiro[5.6]dodecane-9-carbonyl}phenyl)-1,3-diazinane-2,4-dione
N3-(1-benzylpiperidin-4-yl)-N5-tert-butyl-1-cyclohexyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
6-fluoro-2-({[(1S,2R)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-yl]amino}methyl)quinolin-4-ol
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
(4aR,8aS)-1-[(3-fluorophenyl)methyl]-6-[3-(4-methylphenyl)propanoyl]-decahydro-1,6-naphthyridin-2-one
1-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5,5-diphenylpiperidin-2-one
2-methoxy-N-(2-methyl-3-{[(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)carbamoyl]amino}phenyl)acetamide
N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2-(2,3,6-trifluorophenyl)acetamide
3-{4-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]-4-oxobutyl}-3,4-dihydroquinazolin-4-one
(2S,4S)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-N-ethyl-4-(1-methylcyclopropaneamido)pyrrolidine-2-carboxamide
6-[1-(4-propylpyrimidine-5-carbonyl)piperidin-3-yl]pyrimidin-4-ol
3-chloro-5-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
2-(1-methyl-1H-pyrrol-2-yl)-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-oxoacetamide
1-[2-({[2-(4-fluorophenyl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
4-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-(2-ethylbutyl)-8-[2-(4-methyl-1H-pyrazol-1-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-methyl-2-({[3-(thiophen-3-yl)-1,2,4-oxadiazol-5-yl]methyl}sulfanyl)-3,4-dihydropyrimidin-4-one
2-[(3-chlorophenyl)methyl]-N-[1-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(4-methylphenyl)ethan-1-one
3-{[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]methyl}-N-(1-methyl-1H-1,2,3-triazol-4-yl)benzamide
methyl (2S,4S)-4-[2-chloro-5-(trifluoromethyl)benzamido]-1-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidine-2-carboxylate
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[3-(trifluoromethoxy)phenyl]methyl}acetamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-2-(2,4-dichlorophenoxy)-N-methylacetamide
2,4-dimethyl-N-[(3R,5S)-1-(3-methylbut-2-en-1-yl)-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]pyrimidine-5-carboxamide
(2S,4S)-4-amino-1-(6-methylquinoline-4-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
6-[2-(ethylamino)pyrimidine-5-carbonyl]-2-methyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
(1S,6R)-3-[(2-chloro-4-fluorophenyl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
3-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-N-[(4-methylphenyl)methyl]propanamide
4-(4-methyl-1H-pyrazol-1-yl)-1-[2-(propan-2-yl)pyrimidine-4-carbonyl]piperidine-4-carboxylic acid
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-(propan-2-yl)-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
({4-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1,4-oxazepan-6-yl}methyl)dimethylamine
1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-4-(prop-2-en-1-yl)-1,4-diazepan-5-one
(4aR,7aS)-1-ethyl-4-(3-oxo-3,4-dihydroquinoxaline-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-phenyl-1H-pyrazol-4-yl)methyl]amine
1-[2-(2-ethyl-1,3-thiazol-4-yl)ethyl]-3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)urea
N,N-bis(2-hydroxyethyl)-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
1-{[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
6-methoxy-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]hexan-1-one
9-(2-methoxypropanoyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{3-[({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]piperidin-1-yl}ethan-1-ol