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[(3R,5R)-1-(1H-indole-6-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-(2-methoxyphenyl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
1-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]-3-(1-methyl-1H-pyrazol-4-yl)urea
3-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1-[4-(2-oxopyrrolidin-1-yl)phenyl]urea
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]piperazine
4,4,4-trifluoro-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]butanamide
2,6-diamino-4-{3-[(dimethylamino)methyl]phenyl}-5,6,7,8-tetrahydroquinoline-3-carbonitrile
3-({5-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-1,2,4-oxadiazol-3-yl}methyl)pyridine
4-hydroxy-N-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-2-phenylpyrimidine-5-carboxamide
(1S,5R)-3-[1-(4-methoxyphenyl)piperidin-4-yl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-benzyl-3-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrrolidine
5-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-N-propylpyrimidin-2-amine
(3S,5R)-N3-(2-acetamidoethyl)-N5-(4-fluorophenyl)-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
N3-benzyl-N5-[2-(3-chlorophenyl)ethyl]-1-(2-methoxyethyl)-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
3-[2-(2-methylpropanesulfonyl)ethyl]-1-[4-(1,3-thiazol-4-yl)phenyl]urea
methyl 3-({[(2-chlorophenyl)methoxy]carbonyl}amino)azepane-1-carboxylate
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-[(3-methylthiophen-2-yl)sulfonyl]piperidine
(2R,3R)-3-(1H-imidazol-1-yl)-1'-(thiophene-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-[(cyclohexylamino)methyl]-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
N,N-dimethyl-2-[(1,2,3,4-tetrahydronaphthalen-2-ylformamido)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-[(4-chlorophenyl)methyl]-4-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperazine
1-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
N-[(5-methoxy-1H-indol-2-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-[(4-methylphenyl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
4-{5-methylthieno[2,3-d]pyrimidin-4-yl}-1H-indole
4-[(2,3-dihydro-1H-inden-2-yl)amino]-1-(2,2-dimethylpropyl)pyrrolidin-2-one
4-[2-(piperidine-1-carbonyl)phenoxy]-1-(thian-4-yl)piperidine
4-ethyl-1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]methanol
2-(2,5-dimethoxyphenyl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]acetamide
(3R,4R)-3-cyclopropyl-4-methyl-1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)pyrrolidin-3-ol
1-{3-[1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]phenyl}imidazolidin-2-one
(4aR,8aS)-6-(2-ethylbutanoyl)-1-[(4-fluorophenyl)methyl]-decahydro-1,6-naphthyridin-2-one
N-benzyl-5-(4-chloro-2-methoxyphenoxymethyl)-N-(cyclopropylmethyl)-1,2-oxazole-3-carboxamide
N-(2-methylpropyl)-1-[(1s,4s)-4-[3-(4-methoxyphenyl)propanamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(3R,4S)-1-[1-(methoxymethyl)cyclobutanecarbonyl]-N,N-dimethyl-4-phenylpyrrolidin-3-amine
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)-1,8-naphthyridine-2-carboxamide
2-[2-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)-1H-pyrrol-1-yl]pyrimidine
(4aS,7aR)-1-[(4-fluoro-3-methylphenyl)methyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
1-cyclopropyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
ethyl 1-[3-(morpholin-4-yl)propyl]-1H-imidazole-2-carboxylate
2-(2-methoxy-5-methylphenyl)-2-[methyl(prop-2-yn-1-yl)amino]acetic acid
1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-(butan-2-yl)-N3-(furan-2-ylmethyl)-N5-[(1-hydroxycyclohexyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(1R,7S)-3-(4-fluoro-2-methylphenyl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[2-(pyridin-3-yloxy)propyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide