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6-[3-(hydroxymethyl)piperidin-1-yl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
4-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]-1-(2-methylpropyl)piperidine
1-({3-[2-(methylsulfanyl)ethyl]-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl}methyl)-1H-1,2,3,4-tetrazole
4-(6-methoxypyridin-3-yl)-6-(pyrrolidin-1-yl)pyrimidin-2-amine
2-{4-[ethyl(methyl)sulfamoyl]-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl}acetic acid
6-{4-[3-(2-chlorophenoxy)azetidin-1-yl]piperidin-1-yl}-9H-purine
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}furan-3-carboxamide
1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2,2-dimethylpropan-1-one
3-(2-hydroxyphenyl)-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-1H-pyrazole-5-carboxamide
N-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methoxybenzamide
3,3-dimethyl-1-[(5-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]urea
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-[4-(quinolin-2-yl)-1H-pyrazol-1-yl]acetamide
2-methyl-6-[(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridine
3-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]phenol
4-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-2-(thiophen-2-yl)-1,3-thiazole
2-(cyclopropylmethyl)-N-[(2-methylphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-(4-fluorophenyl)-2-(furan-2-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
3-[(3R,4S)-1-[(2,5-dimethylphenyl)carbamoyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N-(2-hydroxypropyl)-N-methyl-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carboxamide
3-methyl-2-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridine
1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
methyl (1R,3S,3aR,6aS)-3-(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)-5-methyl-1-(2-methylpropyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
ethyl 4-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]piperazine-1-carboxylate
1-(2-methoxyethyl)-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine
1-methyl-2-oxo-8-(1,3-thiazol-2-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-tert-butyl-4-[({[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]pyrrolidin-2-one
2-[6-chloro-3-(piperidin-1-ylmethyl)imidazo[1,2-a]pyridine-2-carbonyl]-1,2,3,4-tetrahydroisoquinoline
1-tert-butyl-N-[2-(4-chlorophenyl)ethyl]-5-oxopyrrolidine-3-carboxamide
N-{2-[4-(1-methylpiperidin-4-yl)morpholin-2-yl]ethyl}cyclopropanesulfonamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(phenylamino)pyrimidine-5-carboxamide
N-cycloheptyl-1-cyclopropyl-4-oxo-5-(4-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-(dimethylamino)-N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-(3-methylphenyl)acetamide
N-({1-[(2,3-dimethoxyphenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
1-benzyl-4-(2-propyl-1,3-thiazole-4-carbonyl)-1,4-diazepan-6-ol
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-propanoylpiperidine-3-carboxamide
5-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-1,2,3-benzotriazole
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
3-chloro-6-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)pyridine-2-carboxylic acid
4-ethyl-6-(4-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperazin-1-yl)pyrimidine
1-[(4-{[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
N-{[3-methyl-7-(1,2,5-thiadiazole-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(phenylsulfanyl)acetamide
1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
2-ethyl-8-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][2-(methylsulfanyl)ethyl]amine
4-(4-fluorophenyl)-1-[2-(methylamino)pyridine-4-carbonyl]piperidin-4-ol
4-ethyl-5-methyl-6-{4-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}pyrimidin-2-amine
2-(3-{[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl}phenoxymethyl)pyridine
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(3-methyl-1H-pyrazol-1-yl)-N-{[7-(methylsulfanyl)-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}propanamide
2-[(3S,4R)-3-acetamido-4-propylpyrrolidin-1-yl]-N-(pyridin-2-ylmethyl)acetamide
4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazine-2-carboxylic acid