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1-[(3-chlorophenyl)methyl]-3-(2-methoxyethyl)-5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-1,2,4-triazole
4-(1-aminocyclopropanecarbonyl)-7-(1,3-benzothiazol-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}-2,1,3-benzothiadiazole
1-[(1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}cyclopropyl)methyl]-1H-pyrazole
2-(2-hydroxyethyl)-9-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
4-(2,2-dimethyl-2,3-dihydro-1-benzofuran-7-yl)-7-(2-oxoimidazolidin-1-yl)-1,2,3,4-tetrahydroquinolin-2-one
{3-[(2-methylphenyl)methyl]-1-(pyridin-2-ylmethyl)piperidin-3-yl}methanol
N4-[2-(dimethylamino)-2-(4-methylphenyl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
(3S,4R)-4-(4-fluorophenyl)-1-(pyrimidin-2-ylmethyl)pyrrolidine-3-carboxylic acid
8-({[(2-methylphenyl)methyl]carbamoyl}methyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
6-methyl-4-(4-methyl-1H-imidazol-5-yl)-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,2,3,4-tetrahydropyrimidin-2-one
2-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-fluoropyridine
(2R,6S)-2,6-dimethyl-4-{5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}morpholine
1-(4-{1-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-1H-imidazol-2-yl}thiophen-2-yl)ethan-1-one
7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
2-(4-ethoxyphenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
{5-[1-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1H-1,2,3-triazol-4-yl]furan-2-yl}methanol
3-{2-[methyl(2-methylpropyl)amino]ethyl}-8-(1-methyl-1H-pyrazole-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[1-(1-{[1,2,4]triazolo[3,4-a]phthalazin-6-yl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-1-ol
N-methyl-5-[({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)methyl]furan-2-carboxamide
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(4-methyl-1,3-oxazole-5-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-(4-cyclopropanecarbonylphenyl)-1-[(4-methoxyphenyl)methyl]-1H-pyrazole
2-methyl-6-[4-oxo-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
8-[5-(2-chlorophenyl)furan-2-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
6-(1,4-diazepan-1-yl)-N2,N2-diethylpyrimidine-2,4-diamine
N-(cyclohex-1-en-1-ylmethyl)-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
N-[(1R,2R)-2-acetamido-2,3-dihydro-1H-inden-1-yl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-[(3-fluorophenyl)methyl]-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{2-[(4-benzylpiperazin-1-yl)methyl]-1,3-oxazole-4-carbonyl}-3-ethylpiperazine
methyl 4-[5-methyl-4-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)-1,3-oxazol-2-yl]benzoate
2-(3,4-dimethoxyphenyl)-2-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}acetic acid
2-amino-8-[4-(1H-imidazol-1-yl)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(pyridin-2-yl)pyrimidine-5-carboxamide
5-(3-fluorophenoxymethyl)-N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-1H-pyrazole-3-carboxamide
1-(3-methoxypropyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
4-{[8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}benzonitrile
N-(1,3-benzothiazol-2-ylmethyl)-5-methoxy-N,1-dimethyl-1H-indole-2-carboxamide
2-hydroxy-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2-[4-(trifluoromethyl)phenyl]acetamide
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(ethyl)(2-methoxyethyl)amine
N-methyl-5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-(pyridin-3-ylmethyl)pyridin-2-amine
N-[(3R,4S)-1-(2-amino-6-methylpyrimidin-4-yl)-4-cyclopropylpyrrolidin-3-yl]-3-methoxy-2,2-dimethylpropanamide
methyl[(2-phenyl-1,3-thiazol-4-yl)methyl][1-(pyridin-4-yl)ethyl]amine
6-methoxy-N-({3-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(pyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
6-ethoxy-3-{[(1S,6R)-3-methyl-3,9-diazabicyclo[4.2.1]nonan-9-yl]methyl}-1,2-dihydroquinolin-2-one
2-{5-[2-amino-6-(cyclopropylamino)pyrimidin-4-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
3-methyl-1-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidine
4-(dimethyl-1,3-thiazole-5-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-methanesulfonylpropan-1-one