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6-(1-{imidazo[1,2-a]pyridin-6-ylmethyl}piperidin-4-yl)-2-(2-methoxyethyl)-3,4-dihydropyrimidin-4-one
N-methyl-2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
3-methyl-2-propyl-4-(quinolin-8-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-{2-[2-(4-fluorophenyl)azetidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
2-{3-cyclopropyl-5-[2-(2-oxo-1,2-dihydropyridin-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
6-cyclopentyl-N-[3-(1H-imidazol-1-yl)propyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(4-ethoxyphenyl)methyl]-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
N-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
6-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-4-oxo-4H-pyran-2-carboxamide
5-[(dimethylamino)methyl]-N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}furan-2-carboxamide
4-(2,3-dihydro-1H-inden-2-yl)-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
{2-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]phenyl}methanol
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
N-[3-({[1-(4-methylpyridin-2-yl)propyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
N-({5-[(3,5-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
(3S,4S)-1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]piperidine-3,4-diol
(2S)-4-methyl-1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-2-(propan-2-yl)piperazine
1-{1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}propan-1-ol
3-(4-methoxyphenyl)-3-phenyl-N-(pyridin-2-ylmethyl)propanamide
6-({[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}amino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N,2-dimethyl-1H-imidazole-4-carboxamide
3-cyclopropyl-4-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]acetamide
N-cyclopropyl-2-phenyl-N-(1,3-thiazol-2-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
1-{3-[7-(3-chlorophenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]phenyl}imidazolidin-2-one
3-{[1-(ethylcarbamoyl)piperidin-4-yl]methyl}benzoic acid
9-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-(1-methylpiperidin-4-yl)pyrrolidine-2-carboxylate
N-methyl-N-[2-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)ethyl]-1-benzothiophene-2-carboxamide
N-ethyl-2-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
N,N,4-trimethyl-3-({[(4-methylpyridin-2-yl)methyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-methyl-4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-2-one
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]pyrrolidin-3-yl]acetamide
3-(hydroxymethyl)-1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-ol
methyl (2S,4S)-1-[(2-hydroxyphenyl)methyl]-4-{2-[3-(trifluoromethyl)phenyl]acetamido}pyrrolidine-2-carboxylate
(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-methylpiperazin-2-yl)methanol
1-[2-(dimethylamino)ethyl]-N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-5-oxopyrrolidine-3-carboxamide
(2R,3R)-3-(azepan-1-yl)-1'-(furan-2-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-[4-(pyrazin-2-yl)piperazin-1-yl]butan-1-one
4-(1-ethyl-1H-imidazol-2-yl)-1-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)piperidine
N-methyl-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-{2-[2-(prop-2-en-1-yl)phenoxy]ethyl}benzamide
1-{[2-(3-methoxypyrazin-2-yl)phenyl]methyl}piperidin-4-one
6-methyl-2-{3-[1-(pyridin-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridine-3-carbonitrile
(2-{[4-(3-methylpyrazin-2-yl)piperazin-1-yl]methyl}phenyl)methanol
4-(1H-pyrazol-3-yl)-N-[2-(4-sulfamoylphenyl)ethyl]benzamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(4-oxo-3,4-dihydro-1,2,3-benzotriazin-3-yl)acetamide
4-[(4-methyl-5-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}-4H-1,2,4-triazol-3-yl)methyl]piperidine
N-{1-[1-(3,3-dimethylcyclohexyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
N-{2-[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}thiophene-2-carboxamide
methyl 2-(2,4,6-trimethylphenyl)pyridine-4-carboxylate