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3-[(3R,4S)-4-(morpholin-4-yl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-3-yl]propanoic acid
3-[2-(dimethylamino)ethyl]-5-[(3-fluorophenyl)methyl]-5-{1-[(2E)-3-phenylprop-2-enoyl]piperidin-4-yl}imidazolidine-2,4-dione
2-(1'-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl)acetamide
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[(1R,2S)-2-phenylcyclopropyl]acetamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-1-(4-methoxyphenyl)-2,2-dimethylcyclopropane-1-carboxamide
7-[3-(morpholine-4-carbonyl)benzenesulfonyl]-1-oxa-7-azaspiro[3.5]nonane
8-{[3-hydroxy-2-oxo-1-(2-phenylethyl)piperidin-3-yl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2,2-dimethyl-N-{2-[4-(pyridin-2-ylmethyl)morpholin-2-yl]ethyl}propanamide
2-(4-{[(butan-2-yl)(pyridin-2-ylmethyl)amino]methyl}phenyl)-5-fluoro-6-methyl-3,4-dihydropyrimidin-4-one
N-cyclopropyl-1-[2-(3,4-dimethoxyphenyl)acetyl]piperazine-2-carboxamide
2-ethoxy-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-methylpropan-1-one
N-cyclopropyl-3-(4-fluorophenyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-phenylpropanamide
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-2-(4-propanoylphenoxy)acetamide
(3-{2-[1-(4-fluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
3-(2H-1,3-benzodioxol-5-yl)-1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]propan-1-one
(1R,2S,6R,7S)-4-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-4-azatricyclo[5.2.2.02,6]undecane
5-ethyl-1'-[(1-ethyl-1H-indol-6-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,3-benzodiazole
1-(2-methyl-1,3-benzothiazol-6-yl)-3-[2-(N-methylmethanesulfonamido)ethyl]urea
(3S,4R)-1-(3-chloro-4-ethoxybenzoyl)-4-methyl-3-(2-methylpropyl)piperidin-4-ol
1-(4-fluorophenyl)-4-{8-methyl-2,8-diazaspiro[4.5]decan-2-yl}butane-1,4-dione
2-methyl-8-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanoyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-[(2-amino-1,3-thiazol-4-yl)methyl]-5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carboxamide
5-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-4-methyl-2-(propan-2-yl)pyrimidine
N-benzyl-N-butyl-3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
2-{3-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]propyl}phenol
1-({5-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-ylmethyl]-2,4-dimethylphenyl}methyl)-4-methylpiperazine
5,6-dimethyl-2-{2-oxo-2-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-2,3-dihydropyridazin-3-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
(3aR,7aS)-5-methyl-2-[6-(piperidin-4-yl)pyrimidin-4-yl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
methyl({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})(pyrazin-2-ylmethyl)amine
3-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)-1-methyl-1,2-dihydroquinoxalin-2-one
(2R,3R,6R)-3-(4-methylphenyl)-5-(pyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-methoxy-N-[(1-methylpiperidin-3-yl)methyl]cyclohexane-1-carboxamide
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
5-{[3-(3-methoxypiperidine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}-2-methyl-1,3-benzothiazole
3-[2-(pyridin-2-yl)-1H-imidazol-1-yl]-N-(1,3-thiazol-2-yl)propanamide
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-[2-(2-methylphenyl)ethyl]piperidine
3-[1-(1-methanesulfonylpyrrolidine-2-carbonyl)azetidin-3-yl]pyridine
1-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]ethan-1-one
(3S,4S)-1-[(5-ethylpyridin-2-yl)methyl]-4-(4-fluorophenyl)piperidin-3-ol
6-[(4-chlorophenyl)methyl]-3-(oxolan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
{2-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}urea
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
4-[1-(3-chloro-4-methylphenyl)piperidin-4-yl]-N-cyclopropylpiperazine-2-carboxamide
2-{4-[1-(2-methoxyethyl)piperidine-3-carbonyl]piperazin-1-yl}benzonitrile
N,N-dimethyl-5-[(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)methyl]pyridin-2-amine
3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
(2S,4S)-4-amino-N,N-diethyl-1-(2-methoxybenzenesulfonyl)pyrrolidine-2-carboxamide