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1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
{[1-(1-cycloheptylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl}diethylamine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-methyl-4-oxo-4H-pyran-2-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]propanamide
6-cyclobutyl-2-(2-{[cycloheptyl(methyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
3-methyl-N-({3-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(1,3-thiazol-4-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
N-[(3S,4R)-4-(propan-2-yl)-1-(pyridine-4-carbonyl)pyrrolidin-3-yl]acetamide
(3S,4S)-4-cyclopropyl-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]pyrrolidine-3-carboxylic acid
4-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-(6-methoxynaphthalen-2-yl)morpholine
5-{[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-3-(propan-2-yl)-1,2,4-oxadiazole
3,6-dimethyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1-benzofuran-2-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
6-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-N,N-dimethylpyrimidin-4-amine
3-chloro-N-methyl-N-(pyrimidin-4-ylmethyl)thiophene-2-carboxamide
4-(2-methoxyphenoxy)-1-[6-methyl-2-(methylamino)pyrimidin-4-yl]piperidine-4-carboxylic acid
N-[2-({[2-methyl-3-(pyrrolidin-1-yl)phenyl]carbamoyl}amino)ethyl]pyridine-3-carboxamide
1-[2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]imidazolidin-2-one
methyl 4-oxo-4-[3-(phenylamino)piperidin-1-yl]butanoate
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]{[6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1H-indazole-3-carboxamide
2-(2-ethyl-1H-imidazol-1-yl)-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]acetamide
N-[2-(4-methoxyphenyl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
(2R)-2-amino-1-{4-[4-(3-hydroxypropyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}hexan-1-one
N-[3-(4-fluorophenyl)phenyl]-1-(oxane-4-carbonyl)piperidine-3-carboxamide
2-[4-(2-ethylpyrimidine-5-carbonyl)piperazin-1-yl]-4-phenylpyrimidine
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[(2-fluorophenyl)methyl]piperidine
2-(2H-1,3-benzodioxol-5-yloxy)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}propanamide
2-[5-(2-chloro-4,5-difluorophenyl)-1-cyclohexyl-1H-1,2,4-triazol-3-yl]acetamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-[2-fluoro-6-(propan-2-yloxy)phenyl]-2-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}acetic acid
1-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-4-methylpiperazine
2-butyl-5-(thiomorpholine-4-carbonyl)-1,3-benzoxazole
(2R,6R)-4-{2-[benzyl(methyl)amino]acetyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(4-hydroxyphenyl)propan-1-one
2-[1-butyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]pyrazine
(1S,5R)-3-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(4-acetylphenoxy)-1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
1-(3-methoxybenzoyl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperazine
5-acetyl-3-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
4-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}morpholine
2-methyl-4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
methyl 4-{4-[(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)methyl]-5-methyl-1,3-oxazol-2-yl}benzoate
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(piperidine-1-carbonyl)pyridine
N-(1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-fluorobenzamide
3-(6-methoxy-3-methyl-1-benzofuran-2-amido)pyrrolidine-3-carboxylic acid
7-(5-phenyl-1,3,4-thiadiazol-2-yl)-2,7-diazaspiro[4.4]nonane-1,3-dione