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3-(ethylsulfanyl)-1-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
4-(4-chlorophenyl)-1-[3-(propoxymethyl)pyrrolidin-1-yl]butan-1-one
5-cyclobutyl-N-[3-(1H-imidazol-1-yl)propyl]-1,3,4-oxadiazol-2-amine
2-[(3,4-difluorophenyl)methyl]-8-[(2S)-3-hydroxy-2-methylpropyl]-2,8-diazaspiro[4.5]decan-3-one
6-[({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)amino]pyridine-2-carbonitrile
4-{3-[2-(2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethyl]morpholine-4-carbonyl}-6-(2-methylpropyl)-1,2-dihydropyrimidin-2-one
2-(azocan-1-yl)-N-{[1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]methyl}acetamide
(2R)-2-amino-N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-4-methylpentanamide
N-ethyl-N-(2-hydroxy-3-phenoxypropyl)-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
3-({4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
N-(1H-indol-2-ylmethyl)-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
4-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]-2,6-dimethylquinoline
5-[2-(3-methoxypropyl)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
2-{4-[(2,5-dimethylphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
1-methyl-2-{2-[3-(1H-pyrazol-1-yl)propyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-1H-1,3-benzodiazole
2-ethyl-9-[1-(4-methylphenyl)cyclopropanecarbonyl]-2,9-diazaspiro[5.5]undecan-3-one
1-({5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propan-2-ol
1-[1-(4-fluorophenyl)cyclopropanecarbonyl]-3-(2-methoxyphenoxy)azetidine
3-({ethyl[(1R,2R)-2-hydroxycyclohexyl]amino}methyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)benzamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-(2-hydroxypropyl)-N-methyl-1,3-oxazole-4-carboxamide
1-(4-methylpiperazin-1-yl)-3-[1-(quinazolin-4-yl)piperidin-3-yl]propan-1-one
N'-benzyl-N'-(4-hydroxybutyl)-N-(4-methylphenyl)propanediamide
2-(4-chlorophenoxy)-1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-(2-methoxyethyl)-3-methyl-N-[(5-methylthiophen-2-yl)methyl]-1H-indole-2-carboxamide
2-{1-[(4-fluorophenyl)methyl]-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
6-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-(1,2-oxazol-5-ylmethyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
2-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-amino-N-[3-(azepan-1-yl)propyl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-methylacetamide
N-[3-(1H-imidazol-1-yl)propyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)[3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl)amine
N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
2-(3-acetyl-1H-indol-1-yl)-N-[(6-oxo-1,6-dihydropyrimidin-4-yl)methyl]butanamide
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(1H-indol-3-yl)acetamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[5-(propan-2-yl)thiophene-3-carbonyl]pyrrolidin-3-yl]methanol
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
1-(2-amino-5-methylpyrimidin-4-yl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
4'-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-{[6-(4-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-4-methyl-1,4-diazepane
N-[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]-2-(dimethylamino)acetamide
1-[(4-fluoro-2-methylphenyl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-(2,3-dihydro-1H-inden-4-yl)-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
6-(pyridin-4-ylmethyl)-5,6-dihydro-1,6-naphthyridin-5-one
6-(4-methylpiperazin-1-yl)-N4-[2-(3-methylthiophen-2-yl)ethyl]pyrimidine-2,4-diamine
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]acetamide
2-[4-(4H-1,2,4-triazol-3-ylmethyl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
(3R,4R)-4-(hydroxymethyl)-1-[5-(3-methoxyphenyl)furan-2-carbonyl]piperidin-3-ol
3-cyclopropyl-1-[2-methoxy-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-[(1-methyl-1H-pyrazol-4-yl)methyl]urea