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[(2-butoxy-3-methoxyphenyl)methyl][1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]amine
methyl({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})(pyridin-2-ylmethyl)amine
methyl 1-{3-carbamoyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-7-carbonyl}cyclopropane-1-carboxylate
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
3-(3-methoxyphenyl)-N-[3-(pyridin-4-yl)propyl]-1H-pyrazole-4-carboxamide
[(2-methyl-1H-imidazol-4-yl)methyl](3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)amine
3-(oxolan-3-yl)-5-[1-(propan-2-yl)-1H-pyrazol-3-yl]-1,2,4-oxadiazole
1-methyl-5-[(3-methylbutyl)amino]-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-4-methoxy-N-methylbenzamide
methyl N-{2-[4-(2-chlorophenoxy)piperidin-1-yl]-2-oxoethyl}carbamate
2-(3-acetyl-1H-pyrazol-1-yl)-N-{1-[(2-methoxyphenyl)methyl]-1H-pyrazol-5-yl}acetamide
3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-cycloheptanecarbonylpiperidine
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(piperidin-1-yl)acetamide
[(3R,5R)-1-(5-chlorothiophene-2-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
8-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
7-[3-(1H-imidazol-5-yl)-2-(1H-pyrrol-1-yl)propanoyl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-[(8-chloroquinolin-2-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
N-[4-(4-{[2-(2-methoxyphenyl)ethyl]amino}piperidin-1-yl)phenyl]-3-phenylpropanamide
(1S,5R)-6-(2-methoxyethyl)-3-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[3-(ethylsulfanyl)phenyl]-6-(piperidine-1-carbonyl)pyrazine
N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(5-methyl-1H-pyrazol-1-yl)acetamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
3-[5-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
ethyl({[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl})(2-methylprop-2-en-1-yl)amine
2-chloro-4-[3-(4-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridine
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrazole-4-carboxamide
(3R,4R)-4-amino-1-({4-methoxy-3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperidin-3-ol
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
(2R,6R)-11-methoxy-4-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]-4-(oxan-4-yl)piperazine-1-carboxamide
2-methoxy-1-{8-[(4-methylpiperazin-1-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}ethan-1-one
3-ethyl-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
4-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
2-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}-5-methoxypyridin-4-ol
1-(cyclopropylmethyl)-5-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(4S)-4-(methoxymethyl)-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-3,3-dimethylpiperidin-4-ol
(3E)-4-phenyl-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]but-3-enoic acid
N-{[7-fluoro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-5-methylthiophene-2-carboxamide
1-[1'-(5-chlorothiophene-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methyl-1H-pyrazole-3-carboxamide
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-2-(thiophene-2-sulfonamido)acetamide
4-[2-(8-methoxyquinolin-2-yl)-1H-imidazol-1-yl]benzene-1-sulfonamide
3-[methyl({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl})amino]-1-phenylpropan-1-ol
7-(cyclopropylmethyl)-2-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-2,7-diazaspiro[4.5]decan-6-one
2-[(1,4-dioxan-2-ylmethyl)(methyl)amino]-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-6-(thiophen-2-yl)pyridine-3-carboxamide
1-[(2,3-dimethoxyphenyl)methyl]-2-(5-methylfuran-2-yl)-1H-imidazole
(1s,4s)-4-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]cyclohexan-1-ol
4-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]pyridin-1-ium-1-olate