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3-chloro-5-[4-(quinazolin-4-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
4-(1H-imidazol-1-ylmethyl)-1-[4-(pyridin-3-yl)pyrimidin-2-yl]piperidin-4-ol
5-{1-[3-(2-methoxyacetamido)benzoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
(3R,5R)-5-(morpholine-4-carbonyl)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]piperidine-3-carboxamide
3-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[2-fluoro-5-(4H-1,2,4-triazol-4-yl)phenyl]urea
2-[(4-chlorophenyl)methyl]-8-[3-(1H-pyrazol-1-yl)propyl]-2,8-diazaspiro[4.5]decan-3-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-7-methyl-2-oxo-1H,2H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
1-[4-(1H-imidazol-1-yl)phenyl]-N-[4-(methylamino)butyl]piperidin-4-amine
N,N-diethyl-4-[(3-methoxypropyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(1H-pyrazole-3-carbonyl)piperazin-2-yl}ethan-1-ol
4-{2-[benzyl(methyl)amino]-2,3-dihydro-1H-indene-2-carbonyl}piperazin-2-one
N-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}ethane-1-sulfonamide
1-methyl-4-({2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
1-cyclopentyl-3-({1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-3-yl}methyl)urea
4-({3-[4-(2-methylpropyl)piperazine-1-carbonyl]-1,2-oxazol-5-yl}methyl)morpholine
3-(3-fluorophenoxymethyl)-1-[3-(1H-pyrazol-1-yl)benzoyl]piperidine
7-(cyclobutylmethyl)-2-(cyclopentylmethyl)-2,7-diazaspiro[4.5]decane
(3aS,6aS)-2-cyclobutanecarbonyl-5-[(3-fluoro-5-methylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{[4-(3-chlorophenyl)-5-({methyl[(5-methylthiophen-2-yl)methyl]amino}methyl)-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
[(3,4-difluorophenyl)methyl]({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amine
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
1-benzyl-4-[(6-methylpyridin-2-yl)methyl]-1,4-diazepan-6-ol
8-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-[ethyl(methyl)amino]propanamide
2-{1-cyclopentyl-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
(2S,4R)-N-ethyl-4-(4-fluorobenzamido)-1-(1H-imidazol-4-ylmethyl)pyrrolidine-2-carboxamide
2,6-dimethyl-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]pyrimidine-4-carboxamide
4-[(3-hydroxypyrrolidin-3-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
2-[2-methyl-4-(3,3,4-trimethylpiperazin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]acetic acid
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-phenylmethanesulfonylpiperidine
N-[(3R,4S)-1-cyclohexyl-4-cyclopropylpyrrolidin-3-yl]-3-(6-oxo-1,6-dihydropyridazin-3-yl)propanamide
5-(3-fluorophenyl)-N-(3-phenylpropyl)-1,2,4-triazin-3-amine
4-[2-(2-{1-benzyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenoxy)ethyl]morpholine
7-methoxy-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-[(4-benzylpiperidin-1-yl)methyl]-N-methyl-N-(1H-pyrazol-3-ylmethyl)-1,2-oxazole-3-carboxamide
4-({4-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]furan-2-yl}methyl)morpholine
6-(methoxymethyl)-2-[3-({methyl[3-(oxolan-2-yl)propyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N,N-dipropyl-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-(4-methylpiperidin-1-yl)-3-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propan-1-one
(1-{furo[3,2-c]pyridin-4-yl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
3-({4-[4-(oxolan-2-ylmethyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
(3R,4S)-1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
2-[(3,4-difluorophenyl)methyl]-8-(thiophen-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
4-methoxy-N-(2-methoxyethyl)-2-({1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)benzamide
{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[1-(pyridin-3-yl)propan-2-yl]amine
(3aR,6aR)-2-cyclopentyl-N-[2-(methylsulfamoyl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-cyclopropyl-N-[2-(1,4-dioxo-1,2,3,4-tetrahydrophthalazin-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-[(2-fluorophenyl)methyl]-7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide