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methyl (2S,4S)-1-methyl-4-[3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamido]pyrrolidine-2-carboxylate
2-(4-{[methyl(1H-pyrazol-3-ylmethyl)amino]methyl}phenoxy)acetic acid
4-[5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carbonyl]-3-propylmorpholine
1-(2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,3-oxazole-4-carbonyl)azocane
1-(2-methylpropyl)-4-[1-(2,2,2-trifluoroethanesulfonyl)pyrrolidin-3-yl]piperidine
1-cyclopropyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-5-oxopyrrolidine-3-carboxamide
4-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine
N-[1-(4-methanesulfonylphenyl)propyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
1-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-3-(2-methoxyphenoxy)azetidine
7-(3-chlorophenyl)-4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}pyridin-2-amine
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-[2-(2,4-difluorophenyl)ethyl]-1-(1H-imidazol-4-ylmethyl)piperidine
9-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
pyridin-2-yl[1-(3,4,7-trimethyl-1H-indole-2-carbonyl)piperidin-4-yl]methanol
(2R,3R)-3-{[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2,3-dimethoxy-N-({1-[(4-methylphenyl)methyl]piperidin-3-yl}methyl)benzamide
2-methoxy-1-[1'-(thiophen-2-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)methanol
5-{2-[2-(aminomethyl)morpholin-4-yl]pyrimidin-4-yl}-2-ethoxybenzoic acid
N-[1-(4-fluorophenyl)-5-oxopyrrolidin-3-yl]-2,6-dimethylquinoline-4-carboxamide
7-(4-chlorophenyl)-2-(3-methylpyridin-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-(2,6-dimethoxypyridin-3-yl)-N,N-dimethylpyridin-2-amine
1-(4-cyanophenyl)-3-methyl-3-[(5-propyl-1H-pyrazol-3-yl)methyl]urea
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-[(naphthalen-2-ylmethyl)amino]pyrrolidine-2-carboxamide
4-[3-(4-fluorophenoxy)azetidine-1-carbonyl]-2,8-dimethylquinoline
(4aS,7aR)-1-(6-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4aS,7aR)-1-[(3-ethoxyphenyl)methyl]-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-6-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
2-[3-(4-phenyl-1H-imidazol-5-yl)phenoxy]ethan-1-ol
2-[(2S)-2-aminopentanoyl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-({5-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
methyl 2-[5-methyl-2-({[1,2,4]triazolo[1,5-a]pyrimidin-2-ylformamido}methyl)-2,3-dihydro-1-benzofuran-7-yl]benzoate
2-(1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
4-{3-[(4-fluorophenyl)amino]piperidine-1-carbonyl}-6-(propan-2-yl)pyrimidin-2-amine
1-methyl-2-oxo-8-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-methyl-2-oxo-8-[(2E)-3-phenylprop-2-en-1-yl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(2-hydroxyethyl)-N-[3-(3-methylphenyl)phenyl]pyrrolidine-1-carboxamide
3-(8-chloro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-1-[2-(morpholin-4-yl)ethyl]urea
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]acetamide
N-methyl-2-(2-oxopyrrolidin-1-yl)-N-[(4-phenoxyphenyl)methyl]propanamide
4-ethyl-1-methyl-3-{[1-(3-phenylbutanoyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{2-[benzyl(methyl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl}-3-methoxypropanamide
9-{imidazo[1,2-a]pyridine-2-carbonyl}-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
(2R)-2-{4-phenyl-5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}propanamide
2-[(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)methyl]-5,8-dimethylquinolin-4-ol
(1S,5R)-3-(2H-1,3-benzodioxole-5-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-{[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
1-methyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3-(thiophen-2-yl)-1H-pyrazole-5-carboxamide
3-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}-1-[4-(thiophen-2-ylmethoxy)phenyl]urea