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3-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1-(3,4-difluorophenyl)-3-methylurea
N-[(3R,4R)-3-hydroxy-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl]pyridine-4-carboxamide
12-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraen-6-one
2-[2-(5-chloro-2-ethoxyphenyl)phenyl]-5-methyl-1,3,4-oxadiazole
2-hydroxy-N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-5-methylbenzamide
methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
1-methyl-9-(2,7,8-trimethylquinoline-4-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
4-(propan-2-yl)-6-{4-[(propan-2-yloxy)methyl]piperidin-1-yl}pyrimidin-2-amine
1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-3-(pyridin-2-yl)propan-1-one
1-(3,5-difluorophenyl)-N-(1H-indol-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-6-chloropyridazin-3-amine
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-cyclopropyl-1-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidine-2-carboxamide
3-methyl-4-[1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)pyrrolidin-2-yl]-1,2,5-oxadiazole
2-[2-({2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)phenoxy]ethan-1-ol
3-{1-[4-(piperidin-3-yl)benzoyl]piperidin-4-yl}phenol
(1R,3S)-3-(2-hydroxyethoxy)-7-(2-methanesulfonylethyl)-7-azaspiro[3.5]nonan-1-ol
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-3-(pyridin-2-yl)propan-1-one
N'-{4-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-N-(2-methylpropyl)ethanediamide
N-[3-(5-chloro-1H-1,3-benzodiazol-2-yl)propyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
(4aS,8aS)-N-[4-(difluoromethoxy)-2-methylphenyl]-4a-hydroxy-decahydroisoquinoline-2-carboxamide
3-{[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}-8-methyl-1,2-dihydroquinolin-2-one
6-(azocan-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
5-(2-chloro-4-fluorophenoxymethyl)-N-(1H-imidazol-2-ylmethyl)-1,2-oxazole-3-carboxamide
1'-[(3-phenyl-1H-pyrazol-4-yl)methyl]-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-methyl-3-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]urea
3-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-1-methyl-1-[3-(1-methyl-1H-imidazol-2-yl)propyl]urea
3-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
2-methyl-8-(piperidine-1-sulfonyl)-2,8-diazaspiro[4.5]decane
(2-methoxyethyl)[(4-methyl-1H-imidazol-5-yl)methyl][(2E)-3-phenylprop-2-en-1-yl]amine
N-(6-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(5-{[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methyl}furan-2-yl)methyl]-N-methylmethanesulfonamide
N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-1H-pyrazole-4-carboxamide
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
3-[2-(3,4-difluorophenyl)acetyl]-N-[(3-fluorophenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N'-[2-(propan-2-yl)phenyl]butanediamide
6-methyl-2-(3-{[3-(pyridin-2-yloxy)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
1-{2-[3-(5-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[(4-methylthiophen-2-yl)sulfonyl]piperidine
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
N-[(3S,4R)-1-(2-fluoro-5-sulfamoylbenzoyl)-4-propylpyrrolidin-3-yl]acetamide
5-[5-(cyclopropylmethyl)-1,2,4-oxadiazol-3-yl]-6-methyl-2-(1-methyl-1H-pyrazole-5-carbonyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
4-(2-{4-[(4-methoxy-2,3,6-trimethylphenyl)methyl]piperazin-1-yl}ethyl)morpholine
1-(butane-1-sulfonyl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-9H-purin-6-amine
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(methylamino)ethan-1-one
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-amine
3-ethyl-1-[2-methyl-3-(pyrrolidin-1-yl)phenyl]-3-(2,2,2-trifluoroethyl)urea
(4aS,7aR)-1-(1H-imidazol-2-ylmethyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
dimethyl(3-{2-[1-(pyrrolidine-1-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine