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4-{[1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]methyl}morpholine
4-chloro-5-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1-methyl-3-(trifluoromethyl)-1H-pyrazole
(2S,4S)-1-benzyl-N-ethyl-4-{[(3-phenoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
6-cyclopentyl-2-methoxy-3-{[(4-methylpentan-2-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
(2S)-2-amino-2-(2-chlorophenyl)-N-propyl-N-(pyridin-3-ylmethyl)acetamide
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine
4-(1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)thiomorpholine
1-[cyclohexyl(methyl)amino]-3-[2-({[2-(pyridin-3-yloxy)ethyl]amino}methyl)phenoxy]propan-2-ol
3-(1,2-oxazinan-2-yl)-1-{3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidin-1-yl}propan-1-one
1-[1-(2,2-dimethylpropyl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
{[2-(2-methylphenoxy)pyridin-3-yl]methyl}({[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl})amine
N-[(3R,4S)-1-[(4-methyl-1,3-thiazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]oxane-4-carboxamide
ethyl 4-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]piperidine-1-carboxylate
2-{2-[2-(4-fluorophenyl)piperidin-1-yl]ethyl}pyridine
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-ylmethyl)acetamide
N-[(3R,4S)-1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-4-(propan-2-yl)pyrrolidin-3-yl]cyclobutanecarboxamide
(1r,4r)-4-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}cyclohexan-1-ol
ethyl 4-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-amido}piperidine-1-carboxylate
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
4-[3-(3-methylphenoxy)azetidin-1-yl]-4-oxobutane-1-sulfonamide
2-(2,4-dimethylphenyl)-2-{4-[(2-methoxyphenyl)methyl]piperazin-1-yl}acetic acid
5-[1-(piperidin-1-yl)ethyl]-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)furan-2-carboxamide
5-(2-{2-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)amino]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
5-acetyl-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}thiophene-2-carboxamide
2-{5-[1-(dimethyl-1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
3-[(3,4-difluorophenyl)amino]-N-(2,6-dimethylphenyl)piperidine-1-carboxamide
N-[2-(4-benzylpiperazin-1-yl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
5-(4-acetyl-2-methoxyphenoxymethyl)-N-[1-(pyridin-4-yl)propyl]-1,2-oxazole-3-carboxamide
2-(2-chloro-4-fluorophenyl)-1-[2-(3-methoxypropyl)piperidin-1-yl]ethan-1-one
ethyl 4-[(3-fluorophenyl)methyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-4-carboxylate
4-({3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1-phenyl-1H-1,2,3-triazole
2-[3-(methylsulfanyl)phenyl]-2-[4-(morpholin-4-yl)piperidin-1-yl]acetic acid
(3S,5S)-5-[(pyridin-2-ylmethyl)carbamoyl]-1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidine-3-carboxylic acid
2,3,5-trimethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
7-cyclohexyl-2-(1H-pyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-(2,1,3-benzothiadiazol-4-yl)-3-phenyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
6-ethyl-N4-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-5-methylpyrimidine-2,4-diamine
7-(cyclobutylmethyl)-2-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
5-{2-cyano-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-methyl-2-(oxan-2-ylmethoxy)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
8-(6-cyclopropylpyrimidin-4-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-cyclohexyl-2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-(prop-2-yn-1-yl)acetamide
N-{2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}-2-(naphthalen-1-yl)acetamide
N-{[1-(4-chlorophenyl)cyclopropyl]methyl}-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
3-{[(3aR,6aR)-2-methyl-octahydropyrrolo[3,4-c]pyrrol-3a-yl]formamido}-N-(2-methoxyphenyl)propanamide
3-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
8-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(azepane-1-carbonyl)-5-[4-(morpholin-4-yl)piperidin-1-yl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole
2-(furan-2-yl)-N-[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]pyrrolidine-1-carboxamide