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ethyl 4-({4-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}methyl)piperazine-1-carboxylate
2-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidine-1-carbonyl}pyridin-3-ol
4-ethyl-1-methyl-3-{1-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(pyrrolidin-1-yl)-5-(4H-1,2,4-triazol-4-yl)benzonitrile
2-{2-[(3,3-diethylpyrrolidin-1-yl)methyl]phenyl}-6-(propan-2-yl)-3,4-dihydropyrimidin-4-one
[(2S,6S)-4-[(3-methyl-1-benzofuran-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
3-(2-oxopyrrolidin-1-yl)-N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]benzamide
N-(2-hydroxyethyl)-2-(morpholin-4-yl)-2-(pyridin-3-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
6-fluoro-4-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
4-(2,4-dioxoimidazolidin-1-yl)-N-[(2-ethoxypyridin-3-yl)methyl]benzamide
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-3-(1-methylpiperidin-3-yl)propanamide
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-4-(4H-1,2,4-triazol-4-yl)benzamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(2-methyl-1H-1,3-benzodiazol-5-yl)formamido]acetic acid
8-[2-(piperazin-1-yl)phenyl]quinoline
N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]morpholine-2-carboxamide
(2S,4S)-4-amino-N-ethyl-1-[1-(methoxymethyl)cyclobutanecarbonyl]pyrrolidine-2-carboxamide
4-[(3-chlorophenyl)methyl]-1-[3-(furan-2-yl)benzoyl]-1,4-diazepan-5-one
5-[4-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1-cyclopentyl-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
1-{3-oxo-3-[2-(3-phenylpropyl)morpholin-4-yl]propyl}piperidin-2-one
5-phenyl-3-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1,2-oxazole
3-ethyl-1-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidine-3-carboxylic acid
1-[(1-propyl-1H-imidazol-2-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(3R,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidin-3-yl]-3-hydroxypropanamide
N-(cyclohex-1-en-1-ylmethyl)-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
1-{3-[2-(2,3-dihydro-1-benzofuran-5-yl)-1H-imidazol-1-yl]propyl}piperidin-3-ol
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2-(1H-1,2,4-triazol-3-yl)benzamide
(2S,4S)-4-({[4-(benzyloxy)phenyl]methyl}amino)-N-ethyl-1-(propan-2-yl)pyrrolidine-2-carboxamide
2-amino-6-(pyridin-2-yl)-4-[2-(thiophen-2-yl)pyrimidin-5-yl]pyridine-3-carbonitrile
N-cyclopropyl-2,4-dioxo-N-(pyridin-3-ylmethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(2R,3R,6R)-5-(2,6-dimethylpyrimidine-4-carbonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(5-{4-[(4-chlorophenyl)methyl]piperazine-1-carbonyl}-1H-1,3-benzodiazol-2-yl)methanol
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
N,8-dimethyl-N-(propan-2-yl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-2-(pyrrolidin-1-yl)pyrimidine-5-carboxamide
4-[4-chloro-2-(3-methoxypiperidine-1-carbonyl)phenoxy]-1-cyclopentylpiperidine
1-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(2S,4R)-1-benzyl-N,N-diethyl-4-[(1-ethylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
N-{[4-(cyclohexylmethyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl]methyl}-N-methylmethanesulfonamide
2-cyclopentyl-9-[2-(4-fluorophenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(thiophen-3-yl)ethan-1-one
2-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]pyridin-3-ol
4-ethyl-1-methyl-3-({1-[(3E)-4-phenylbut-3-enoyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
1-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2,5-dimethoxyphenyl)ethan-1-one
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-[(3-fluorophenyl)methyl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
N-(2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-oxoethyl)methanesulfonamide
1-{[3-(3-carboxyphenyl)piperidin-1-yl]sulfonyl}piperidine-4-carboxylic acid
5-{2-[8-(2-hydroxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(3,4-dimethoxyphenyl)-5-fluoro-1-[1-(4-methoxybenzoyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-phenyl-1-(2-propoxybenzoyl)piperidin-3-amine