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4-(4-chlorophenoxy)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-4-carboxamide
2-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-4-(3,3,3-trifluoropropyl)pyrimidine
2-(5-methyl-1H-indol-3-yl)pyridine-3-carboxamide
1-[5-(methoxymethyl)-1,3,4-oxadiazole-2-carbonyl]azonane
3-[(3R,4S)-4-(morpholin-4-yl)-1-[5-(pyrrolidin-1-ylmethyl)pyridin-2-yl]piperidin-3-yl]propanoic acid
7-(cyclobutylmethyl)-2-[6-(dimethylamino)pyridine-3-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
(2E)-N-{[3-methyl-7-(quinoxaline-6-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-phenylprop-2-enamide
(3aS,6aS)-2-methyl-5-[2-(4H-1,2,4-triazol-4-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(8R,9aS)-2-[(3,5-dimethoxyphenyl)methyl]-8-hydroxy-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
[1-(4-methoxy-3-methylbenzoyl)-3-propylpiperidin-3-yl]methanol
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-phenylethan-1-one
3-butyl-4-(4-ethyl-5-methylthiophene-3-carbonyl)-1-methylpiperazin-2-one
2-[3,5-dimethyl-4-(quinoline-8-sulfonamido)-1H-pyrazol-1-yl]acetic acid
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]cyclopropanecarboxamide
1-ethyl-3-(hydroxymethyl)-N-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)thieno[2,3-d]pyrimidin-4-amine
(3S,9aR)-3-(2-methylpropyl)-8-[(1-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
N-[1-(azepan-1-yl)-2-methylpropan-2-yl]-2-(dimethylamino)-2-(2-fluorophenyl)acetamide
N-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]-2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
3-benzyl-4-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)piperazin-2-one
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-(oxan-4-yl)pyrrolidine-2-carboxamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(1-phenylethyl)-1,2-oxazole-5-carboxamide
4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{4-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-4-amine
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-(7-fluoro-1H-indol-1-yl)acetamide
5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
2-{5-[1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
1-[(1-{6-[3-(hydroxymethyl)phenyl]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
N-methyl-2-(N-methyl-1-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-3-yl}formamido)acetamide
5-(2-methoxyacetamido)-N-[(3S)-2-oxoazepan-3-yl]-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
2-ethyl-7-(2-methoxybenzamido)-1-methyl-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(3-hydroxypyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[4-(4-{[(2,6-difluorophenyl)formamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-5-(methoxymethyl)furan-2-carboxamide
1-methyl-N-[3-(morpholin-4-yl)propyl]-3-propyl-1H-pyrazole-5-carboxamide
3-[5-oxo-3-(pyrazin-2-yl)-4,5-dihydro-1H-1,2,4-triazol-4-yl]propanoic acid
1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-2-methyl-4-(2-methylphenyl)piperazine
1-(4-chlorophenyl)-N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}cyclopropane-1-carboxamide
3-(4-methoxy-3,5-dimethylbenzoyl)-1-(5-methoxyfuran-2-carbonyl)piperidine
2-methoxy-1-{4-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-one
2-({3-azaspiro[5.5]undecan-9-yl}amino)-2-phenylethan-1-ol
N-{3-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-oxopropyl}acetamide
1-(5-propyl-1,3,4-oxadiazol-2-yl)-4-(thiophene-2-carbonyl)piperazine
2-cyclopropyl-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)acetamide
1-[(2-methoxyphenyl)methyl]-N-methyl-6-oxo-N-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
2-(1H-imidazol-2-yl)-1-[2-(propylsulfanyl)phenyl]-1H-imidazole
[(1-cyclopentylpiperidin-4-yl)methyl][(5-ethylfuran-2-yl)methyl](oxolan-2-ylmethyl)amine
(4aS,7aR)-1-(2-methylpropanoyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione